SCHEMBL1055019

SCHEMBL1055019

O=c1ccc2ccc(-n3ccnc3)cc2n1-c1nc2ccccc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.46
CYP11B2 P19099 2/20 0.46
CYP19A1 P11511 1/20 0.46
AURKA O14965 8/20 0.45
CBFB Q13951 1/20 0.45
FGFR1 P11362 1/20 0.44
FLT1 P17948 1/20 0.44
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
KDM4E B2RXH2 2/20 0.40
ALKBH3 Q96Q83 2/20 0.40
NPC1 O15118 1/20 0.40
CASP3 P42574 1/20 0.40
RAB9A P51151 1/20 0.40
SENP8 Q96LD8 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
SENP6 Q9GZR1 1/20 0.40
NCOA3 Q9Y6Q9 1/20 0.40
PGR P06401 1/20 0.40
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3501399 0.83 AURKA (0.42) CYP11B1CYP11B2CYP19A1AURKACBFB
SCHEMBL1054292 0.77 AURKA (0.64) AURKAKDM4EALKBH3NPC1RAB9A
SCHEMBL1054586 0.77 AURKA (0.53) AURKAKDM4EALKBH3NPC1RAB9A
SCHEMBL1052301 0.77 AURKA (0.69) AURKAKDM4EALKBH3NPC1RAB9A
SCHEMBL4107024 0.75 BCHE (0.49) CYP11B1CYP11B2CYP19A1AURKACBFB
SCHEMBL3502120 0.74 AURKA (0.53) AURKAKDM4EALKBH3NPC1RAB9A
SCHEMBL3501837 0.74 AURKA (0.50) AURKAKDM4EALKBH3RAB9AMEN1
SCHEMBL1054750 0.74 KDM4E (0.56) AURKAKDM4EALKBH3NPC1RAB9A
SCHEMBL3500883 0.71 AURKA (0.64) AURKAKDM4EALKBH3NPC1RAB9A
SCHEMBL4305932 0.71 AURKA (0.52) AURKAKDM4EALKBH3NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7875624-B2 administering a cancer patient 4-amino-5-fluoro-3-[6-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]quinolin-2(1H)-one in the treatment of disorders relating to cell adhesion and metastatic processes; for monitoring the effects of drug by measuring the levels of ICAM, VCAM, or E-selectin in the patient NOVARTIS VACCINES AND DIAGNOSTICS, INC. (US) 2011-01-25 US disclosed
US-20050239825-A1 Modulation of inflammatory and metastatic processes CHIRON CORPORATION 2005-10-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050239825-A1 Modulation of inflammatory and metastatic processes VCAM1, EPCAM, ICAM1 CYP11B1 439/4885CYP11B2 347/4885CYP19A1 3944/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.