SCHEMBL10553045

SCHEMBL10553045

[Li]c1cc2cnccc2n1C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 10/20 0.39
GABRG2 P18507 2/20 0.38
GABRB3 P28472 2/20 0.38
GABRA5 P31644 2/20 0.38
NR1H3 Q13133 3/20 0.37
GPR119 Q8TDV5 2/20 0.36
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRA2 P47869 1/20 0.36
GABRA6 Q16445 1/20 0.36
NAMPT P43490 2/20 0.36
TTK P33981 2/20 0.35
AURKA O14965 1/20 0.35
CDK2 P24941 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6508596 0.85 NR1H2 (0.39) NR1H2GABRG2GABRB3GABRA5NR1H3
SCHEMBL21146832 0.84 GABRG2 (0.43) NR1H2GABRG2GABRB3GABRA5NR1H3
SCHEMBL10552835 0.83 NR1H2 (0.40) NR1H2GABRG2GABRB3GABRA5NR1H3
SCHEMBL18437161 0.82 NR1H2 (0.37) NR1H2GABRG2GABRB3GABRA5NR1H3
SCHEMBL18848182 0.82 NR1H2 (0.40) NR1H2GABRG2GABRB3GABRA5NR1H3
SCHEMBL4037148 0.82 CYP2A6 (0.38) NR1H2GABRG2GABRB3GABRA5NR1H3
SCHEMBL27108521 0.81 NR1H2 (0.46) NR1H2GABRG2GABRB3GABRA5NR1H3
SCHEMBL4725709 0.80 NR1H2 (0.52) NR1H2NR1H3
SCHEMBL4795293 0.80 NR1H2 (0.57) NR1H2NR1H3
SCHEMBL20435588 0.80 NR1H2 (0.36) NR1H2GABRG2GABRB3GABRA5NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4831144-A 1H-pyrrolo [3,2-c]pyrrolidines protected in 1-position useful as intermediates SANOFI (FR) 1989-05-16 US claimed
US-4831032-A CARDIOVASCULAR DISORDERS, HYPOTENSIVE, ISOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1989-05-16 US disclosed
US-4831144-A 1H-pyrrolo [3,2-c]pyrrolidines protected in 1-position useful as intermediates SANOFI (FR) 1989-05-16 US disclosed