SCHEMBL1055459

SCHEMBL1055459

CC1CC(=O)N(C(CCCC(=O)O)C(=O)O)C1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.45
MME P08473 1/20 0.45
CYP2C19 P33261 1/20 0.45
PPM1B O75688 1/20 0.44
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
GLA P06280 1/20 0.38
POLB P06746 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
HPGD P15428 1/20 0.38
ALOX12 P18054 1/20 0.38
NFKB1 P19838 1/20 0.38
APEX1 P27695 1/20 0.38
MAPK1 P28482 1/20 0.38
HSD17B10 Q99714 1/20 0.38
FOLH1 Q04609 3/20 0.35
SMN1; SMN2 Q16637 1/20 0.32
PTGER4 P35408 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16202455 0.81 CYP1A2 (0.43) CYP1A2MMECYP2C19PPM1BKDM4E
SCHEMBL8818955 0.80 MME (0.42) CYP1A2MMECYP2C19PPM1BKDM4E
SCHEMBL8818604 0.79 CYP2C19 (0.44) CYP1A2MMECYP2C19PPM1BKDM4E
SCHEMBL16202433 0.78 MME (0.48) CYP1A2MMECYP2C19PPM1BALDH1A1
SCHEMBL14674752 0.77 ALDH1A1 (0.50) CYP1A2CYP2C19PPM1BKDM4EALDH1A1
SCHEMBL3622599 0.75 MME (0.40) CYP1A2MMECYP2C19PPM1BKDM4E
SCHEMBL5142303 0.75 MME (0.40) CYP1A2MMECYP2C19PPM1BKDM4E
SCHEMBL2325576 0.75 MME (0.40) CYP1A2MMECYP2C19PPM1BKDM4E
SCHEMBL16202440 0.75 MME (0.41) CYP1A2MMECYP2C19
SCHEMBL14357696 0.74 MME (0.45) CYP1A2MMECYP2C19PPM1BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3171171-B1 RECOMBINANT DEAMIDATED GLIADIN ANTIGEN BIO RAD LABORATORIES (US) 2018-07-18 EP claimed
EP-2788760-B1 RECOMBINANT DEAMIDATED GLIADIN ANTIGEN BIO RAD LABORATORIES INC (US) 2017-02-15 EP claimed
EP-2478049-B1 A POLYMER SUPPORT UNIV CAPE TOWN (ZA) 2015-02-25 EP claimed
EP-2659901-B1 Recombinant deamidated gliadin antigen BIO RAD LABORATORIES (US) 2015-01-21 EP claimed
EP-2276499-B1 RECOMBINANT DEAMIDATED GLIADIN ANTIGEN BIO RAD LABORATORIES (US) 2013-06-12 EP claimed
US-7538092-B2 Pharmaceutically active oligosaccharide conjugates FRESENIUS KABI DEUTSCHLAND GMBH (DE) 2009-05-26 US claimed
EP-1549350-B1 PHARMACEUTICALLY ACTIVE OLIGOSACCHARIDE CONJUGATES FRESENIUS KABI DE GMBH (DE) 2008-09-24 EP claimed
US-20060100163-A1 Pharmaceutically active oligosaccharide conjugates FRESENIUS KABI DEUTSCHLAND GMBH (DE) 2006-05-11 US claimed
EP-1549350-A1 PHARMACEUTICALLY ACTIVE OLIGOSACCHARIDE CONJUGATES Fresenius Kabi Deutschland GmbH (DE) 2005-07-06 EP claimed
WO-2004032971-A1 PHARMACEUTICALLY ACTIVE OLIGOSACCHARIDE CONJUGATES FRESENIUS KABI DEUTSCHLAND GMBH (DE) 2004-04-22 WO claimed
EP-1480681-B1 COUPLING LOW-MOLECULAR SUBSTANCES TO A MODIFIED POLYSACCHARIDE FRESENIUS KABI DE GMBH (DE) 2011-04-20 EP disclosed
EP-2269655-A2 Coupling of low molecular weight substances to hydroxyalkyl starch Fresenius Kabi Deutschland GmbH (DE) 2011-01-05 EP disclosed
US-7538092-B2 Pharmaceutically active oligosaccharide conjugates FRESENIUS KABI DEUTSCHLAND GMBH (DE) 2009-05-26 US disclosed
EP-1549350-B1 PHARMACEUTICALLY ACTIVE OLIGOSACCHARIDE CONJUGATES FRESENIUS KABI DE GMBH (DE) 2008-09-24 EP disclosed
US-20060100163-A1 Pharmaceutically active oligosaccharide conjugates FRESENIUS KABI DEUTSCHLAND GMBH (DE) 2006-05-11 US disclosed
EP-1480682-A1 COUPLING PROTEINS TO A MODIFIED POLYSACCHARIDE Biotechnologie Gesellschaft Mittelhessen MBH (DE) 2004-12-01 EP disclosed
EP-1480681-A2 COUPLING LOW-MOLECULAR SUBSTANCES TO A MODIFIED POLYSACCHARIDE Biotechnologie Gesellschaft Mittelhessen MBH (DE) 2004-12-01 EP disclosed
WO-2004032971-A1 PHARMACEUTICALLY ACTIVE OLIGOSACCHARIDE CONJUGATES FRESENIUS KABI DEUTSCHLAND GMBH (DE) 2004-04-22 WO disclosed
WO-2003074088-A2 COUPLING LOW-MOLECULAR SUBSTANCES TO HYDROXYALKYL STARCH BIOTECHNOLOGIE - GESELLSCHAFT MITTELHESSEN MBH (DE) 2003-09-12 WO disclosed
WO-2003074087-A1 COUPLING PROTEINS TO A MODIFIED POLYSACCHARIDE BIOTECHNOLOGIE - GESELLSCHAFT MITTELHESSEN MBH (DE) 2003-09-12 WO disclosed