SCHEMBL10558384

SCHEMBL10558384

COc1ccc(OCCCN2CCC(C(c3ccc(F)cc3)c3ccc(F)cc3)CC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.53
HTR1A P08908 1/20 0.53
DRD2 P14416 1/20 0.53
DRD1 P21728 1/20 0.53
DRD5 P21918 1/20 0.53
DRD3 P35462 1/20 0.53
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
USP2 O75604 1/20 0.52
ALDH1A1 P00352 1/20 0.52
HPGD P15428 1/20 0.52
LMNA P02545 1/20 0.50
HTT P42858 1/20 0.50
HRH3 Q9Y5N1 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10460536 0.94 HTR2A (0.58) HTR2AHTR1ADRD2DRD1DRD5
SCHEMBL10556534 0.94 KMT2A (0.58) DRD2KMT2AMEN1ALDH1A1HRH3
SCHEMBL10461614 0.92 HTR2A (0.47) HTR2AHTR1ADRD2DRD1DRD5
Fumaric Acid SCHEMBL10461600 0.91 HTR2A (0.53) HTR2AKMT2A
Fumaric Acid SCHEMBL10461598 0.91 HTR2A (0.53) HTR2AKMT2A
SCHEMBL10459423 0.89 HRH3 (0.56) KMT2AALDH1A1HRH3
SCHEMBL10563296 0.88 HTR2A (0.53) HTR2AHTR1ADRD2DRD1DRD5
SCHEMBL10560025 0.88 DRD2 (0.69) HTR2AHTR1ADRD2DRD1DRD5
SCHEMBL10559724 0.88 HTR2A (0.56) HTR2AHTR1ADRD2DRD1DRD5
Water SCHEMBL10461590 0.88 HRH3 (0.55) KMT2AALDH1A1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4810713-A Arylalkyl-heterocyclic amines, n-substituted by aryloxyalkyl groups used in a method for allergy treatment A. H. ROBINS COMPANY, INCORPORATED (US) 1989-03-07 US claimed
EP-0235463-A2 N-substituted-arylalkyl and arylalkylene piperidines as cardiovascular antihistaminic and antisecretory agents A.H. ROBINS COMPANY, INCORPORATED (a Delaware corporation) (US) 1987-09-09 EP claimed