SCHEMBL10558447

SCHEMBL10558447

COc1ccc(CC(C)CN)cc1OC

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.58
KDM4E B2RXH2 1/20 0.58
LDHA P00338 1/20 0.56
ALOX15 P16050 2/20 0.55
ALOX12 P18054 2/20 0.55
CA2 P00918 1/20 0.55
CYP19A1 P11511 1/20 0.50
FOS P01100 1/20 0.49
TTR P02766 1/20 0.49
JUN P05412 1/20 0.49
NR3C1 P04150 1/20 0.49
HSD17B1 P14061 1/20 0.49
HSD17B2 P37059 1/20 0.49
AOC3 Q16853 1/20 0.47
ALDH1A1 P00352 1/20 0.47
PPARG P37231 1/20 0.47
PPARD Q03181 1/20 0.47
PPARA Q07869 1/20 0.47
STAT3 P40763 1/20 0.46
POLB P06746 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4060504 0.86 KDM4E (0.59) ATMKDM4ELDHAALOX15ALOX12
SCHEMBL23966140 0.84 LDHA (0.57) ATMKDM4ELDHAALOX15ALOX12
SCHEMBL16973582 0.83 LDHA (0.53) ATMKDM4ELDHAALOX15ALOX12
SCHEMBL9026890 0.82 LDHA (0.60) ATMKDM4ELDHAALOX15ALOX12
SCHEMBL5494607 0.82 LDHA (0.60) ATMKDM4ELDHAALOX15ALOX12
SCHEMBL10437147 0.82 KDM4E (0.58) ATMKDM4ELDHAALOX15ALOX12
SCHEMBL2564908 0.81 LDHA (0.59) ATMKDM4ELDHAALOX15ALOX12
SCHEMBL3371646 0.81 LDHA (0.59) ATMKDM4ELDHAALOX15ALOX12
SCHEMBL31545527 0.81 LDHA (0.59) ATMKDM4ELDHAALOX15ALOX12
SCHEMBL31545634 0.81 LDHA (0.59) ATMKDM4ELDHAALOX15ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4853383-A β-blocking substituted imidazoles MERCK & CO., INC. (US) 1989-08-01 US disclosed
US-4642311-A β-adrenergic blocking imidazolylphenoxy propanolamines MERCK & CO., INC. (US) 1987-02-10 US disclosed
US-4567276-A HYPOTENSIVE AGENTS, ADRENERGIC BLOCKING AGENTS MERCK & CO., INC. (US) 1986-01-28 US disclosed
US-4440774-A ANTIHYPERTENSIVE AGENTS AND B-ANDRENERGIC BLOCKING AGENTS MERCK & CO., INC. (US) 1984-04-03 US disclosed