SCHEMBL10567412

SCHEMBL10567412

Nc1nc(-c2ccccc2)cc(N2CC2)n1

nearest known ligand 0.85

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 5/20 0.85
HTR3A P46098 1/20 0.85
USP2 O75604 1/20 0.85
LMNA P02545 1/20 0.85
TSHR P16473 1/20 0.85
HTT P42858 1/20 0.85
HSD17B10 Q99714 1/20 0.85
ADORA2A P29274 1/20 0.63
ADORA1 P30542 1/20 0.63
HPGD P15428 1/20 0.59
HTR1A P08908 1/20 0.58
ADRA2A P08913 1/20 0.58
ADRA2C P18825 1/20 0.58
HTR1D P28221 1/20 0.58
HTR2A P28223 1/20 0.58
HTR2C P28335 1/20 0.58
HTR7 P34969 1/20 0.58
HRH3 Q9Y5N1 1/20 0.58
KMT2A Q03164 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2167865 0.92 HRH4 (1.00) HRH4HTR3AUSP2LMNATSHR
SCHEMBL2166566 0.90 HRH4 (0.94) HRH4HTR3AUSP2LMNATSHR
SCHEMBL27927184 0.89 USP2 (0.74) HRH4HTR3AUSP2LMNATSHR
SCHEMBL2166919 0.84 HRH4 (0.85) HRH4HTR3AUSP2LMNATSHR
Hydrochloric Acid SCHEMBL603952 0.83 HRH4 (0.82) HRH4HTR3AUSP2LMNATSHR
Hydrochloric Acid SCHEMBL6508476 0.83 LMNA (0.65) HRH4HTR3AUSP2LMNATSHR
SCHEMBL602911 0.82 HRH4 (0.65) HRH4HTR3AUSP2LMNATSHR
SCHEMBL2165190 0.81 HRH4 (0.80) HRH4HTR3AUSP2LMNATSHR
Hydrochloric Acid SCHEMBL604845 0.81 HRH4 (0.64) HRH4HTR3AUSP2LMNATSHR
SCHEMBL27927181 0.80 HRH4 (0.61) HRH4HTR3AUSP2LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4795812-A ANTITUMOR THE UPJOHN COMPANY (US) 1989-01-03 US disclosed
EP-0210228-A1 4-SUBSTITUTED-6-ARYL PYRIMIDINE COMPOUNDS THE UPJOHN COMPANY (US) 1987-02-04 EP disclosed
WO-1986004583-A1 4-SUBSTITUTED-6-ARYL PYRIMIDINE COMPOUNDS THE UPJOHN COMPANY (US) 1986-08-14 WO disclosed