SCHEMBL10568378

SCHEMBL10568378

Cc1csc(-c2ccsc2-c2ccc(F)cc2)c1

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.54
PTGS1 P23219 11/20 0.51
PTGS2 P35354 10/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10567394 0.88 MAPK14 (0.54) MAPK14PTGS1PTGS2
SCHEMBL10567547 0.78 PTGS2 (0.52) MAPK14PTGS1PTGS2
SCHEMBL6050629 0.78 PTGS2 (0.49) MAPK14PTGS1PTGS2
SCHEMBL10843937 0.75 MAPK14 (0.79) MAPK14PTGS1PTGS2
SCHEMBL10954902 0.73 MAPK14 (0.51) MAPK14PTGS1PTGS2
SCHEMBL10909626 0.73 PTGS2 (0.39) MAPK14PTGS1PTGS2
SCHEMBL6050640 0.72 PTGS2 (0.52) MAPK14PTGS1PTGS2
SCHEMBL7833395 0.72 PTGS2 (0.52) MAPK14PTGS1PTGS2
SCHEMBL14922922 0.71 NISCH (0.39)
SCHEMBL18516555 0.71 ESR1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4820827-A 2,3-diaryl-5-bromothiophene compounds of use for the treatment of inflammaton and dysmenorrhea E. I. DU PONT DE NEMOURS AND COMPANY (US) 1989-04-11 US disclosed