SCHEMBL10587100

SCHEMBL10587100

C=C[C@@]1(C)CC(=O)[C@]2(O)[C@@]3(C)[C@@H](O)CCC(C)(C)[C@@H]3[C@H](OC(=O)CN3CCCCC3)[C@H](OC(=O)N(CC)CC)[C@@]2(C)O1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADCY1 Q08828 14/20 0.64
MAPK1 P28482 5/20 0.62
CYP3A4 P08684 4/20 0.62
TSHR P16473 3/20 0.62
NR1I2 O75469 2/20 0.62
ADRA1A P35348 2/20 0.62
CYP2C19 P33261 2/20 0.62
KMT2A Q03164 2/20 0.62
MLNR O43193 1/20 0.62
KCNH2 Q12809 1/20 0.62
MEN1 O00255 1/20 0.62
ALDH1A1 P00352 1/20 0.62
CYP2C9 P11712 1/20 0.62
GMNN O75496 1/20 0.57
BLM P54132 1/20 0.57
PMP22 Q01453 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
CYP2D6 P10635 1/20 0.57
NFKB1 P19838 1/20 0.57
HIF1A Q16665 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10584116 0.99 ADCY1 (0.64) ADCY1MAPK1CYP3A4TSHRNR1I2
SCHEMBL2231230 0.90 ADCY1 (0.77) ADCY1MAPK1CYP3A4TSHRNR1I2
SCHEMBL9583128 0.89 ADCY1 (0.76) ADCY1MAPK1CYP3A4TSHRNR1I2
Hydrochloric Acid SCHEMBL10585966 0.89 ADCY1 (0.65) ADCY1MAPK1CYP3A4TSHRNR1I2
Hydrochloric Acid SCHEMBL10696571 0.89 ADCY1 (0.75) ADCY1MAPK1CYP3A4TSHRNR1I2
SCHEMBL10585512 0.89 MAPK1 (0.59) ADCY1MAPK1CYP3A4TSHRNR1I2
Hydrochloric Acid SCHEMBL10764005 0.89 ADCY1 (0.75) ADCY1MAPK1CYP3A4TSHRNR1I2
SCHEMBL10584035 0.89 ADCY1 (0.52) ADCY1MAPK1CYP3A4TSHRNR1I2
SCHEMBL10763687 0.89 ADCY1 (0.75) ADCY1MAPK1CYP3A4TSHRNR1I2
Hydrochloric Acid SCHEMBL10586061 0.88 MAPK1 (0.58) ADCY1MAPK1CYP3A4TSHRNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0315097-A2 Acyl labdane derivatives, process for their preparation and their use as medicines HOECHST AKTIENGESELLSCHAFT (DE) 1989-05-10 EP disclosed