SCHEMBL1059707

SCHEMBL1059707

C=C[CH]c1ccc(C)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.48
RAB9A P51151 2/20 0.46
NPC1 O15118 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TDP1 Q9NUW8 3/20 0.44
ACHE P22303 2/20 0.44
NFE2L2 Q16236 2/20 0.42
MAPT P10636 2/20 0.39
RELA Q04206 1/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
RECQL P46063 1/20 0.39
MDM2 Q00987 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CA1 P00915 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10650014 0.85 ALDH1A1 (0.50) TDP1ALDH1A1
(E)-1,2-Di-P-Tolylethene SCHEMBL6480905 0.82 CYP2A6 (0.58) CYP2A6RAB9ANPC1SMN1; SMN2TDP1
Butadiene SCHEMBL5137794 0.78 ALDH1A1 (0.61) CYP2A6RAB9ANPC1SMN1; SMN2TDP1
SCHEMBL14911 0.77
SCHEMBL679555 0.77 ALDH1A1 (0.69) CYP2A6RAB9ANPC1SMN1; SMN2TDP1
Ethane SCHEMBL23051531 0.74 ALDH1A1 (0.65) CYP2A6RAB9ANPC1SMN1; SMN2TDP1
Hydrochloric Acid SCHEMBL9861453 0.74 ALDH1A1 (0.65) CYP2A6RAB9ANPC1SMN1; SMN2TDP1
Hydrochloric Acid SCHEMBL9861440 0.74 ALDH1A1 (0.65) CYP2A6RAB9ANPC1SMN1; SMN2TDP1
Ammonia Solution, Strong SCHEMBL9397572 0.74 ALDH1A1 (0.65) CYP2A6RAB9ANPC1SMN1; SMN2TDP1
Ethylene SCHEMBL10713150 0.74 ALDH1A1 (0.65) CYP2A6RAB9ANPC1SMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4347365-A ANTICONVULSANTS, MUSCLE RELAXANTS, SEDATIVES HOFFMANN-LA ROCHE INC. (US) 1982-08-31 US claimed
US-4347364-A INTERMEDIATES THEREFOR HOFFMANN-LA ROCHE INC. (US) 1982-08-31 US claimed
WO-2014170343-A1 DEPOLARIZING AGENTS AND NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS FOR TREATING DOPAMINERGIC-RELATED DISORDERS ICM (INSTITUT DU CERVEAU ET DE LA MOELLE ÉPINIÈRE) (FR) 2014-10-23 WO disclosed
CN-102786454-A Bis[1-aryl(alkyl) substituted allyl]sulphane compound and synthetic method and application thereof UNIV TONGJI 2012-11-21 CN disclosed
US-20120202877-A1 ANTI-INFLUENZA AGENTS GRIFFITH UNIVERSITY (AU) 2012-08-09 US disclosed
EP-2454248-A1 ANTI -INFLUENZA AGENTS Griffith University (AU) 2012-05-23 EP disclosed
WO-2011006208-A1 ANTI -INFLUENZA AGENTS GRIFFITH UNIVERSITY (AU) 2011-01-20 WO disclosed
EP-2152272-A2 NOVEL 2,3-DIAMINO-QUINAZOLINONE DERIVATIVES AND THEIR MEDICAL USE NeuroSearch A/S (DK) 2010-02-17 EP disclosed
WO-2008142140-A2 NOVEL 2,3-DIAMINO-QUINAZOLINONE DERIVATIVES AND THEIR MEDICAL USE NEUROSEARCH A/S (DK) 2008-11-27 WO disclosed
EP-1995016-A1 WATER-DISPERSED FLUX COMPOSITION, ELECTRONIC CIRCUIT BOARD WITH ELECTRONIC COMPONENT, AND THEIR PRODUCTION METHODS Toeikasei Co., Ltd. (JP) 2008-11-26 EP disclosed
EP-0216299-A1 Quinoxaline derivatives, method for their preparartion and their use to protect cultivated plants against phytotoxical reaction of herbicides BASF Aktiengesellschaft (DE) 1987-04-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120202877-A1 ANTI-INFLUENZA AGENTS NEU1, NEU3, NEU4 CYP2A6 1204/4885RAB9A 766/4885NPC1 1219/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.