SCHEMBL10600016

SCHEMBL10600016

C=CCC([O])(OC)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.49
TSHR P16473 2/20 0.49
HTT P42858 1/20 0.46
MAPK1 P28482 1/20 0.42
KMT2A Q03164 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
MEN1 O00255 2/20 0.40
CES1 P23141 1/20 0.37
MAPT P10636 2/20 0.37
KCNN4 O15554 1/20 0.36
ALOX15 P16050 2/20 0.35
ATM Q13315 1/20 0.35
CYP3A4 P08684 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
TP53 P04637 1/20 0.32
ALOX12 P18054 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8837021 0.77 ALDH1A1 (0.47) ALDH1A1TSHRHTTMAPK1KMT2A
SCHEMBL9308834 0.76 CES1 (0.41) ALDH1A1MAPK1KMT2AMEN1CES1
Water SCHEMBL1986090 0.76 ALDH1A1 (0.46) ALDH1A1TSHRHTTMAPK1KMT2A
SCHEMBL11775673 0.74 ALDH1A1 (0.57) ALDH1A1TSHRHTTMAPK1KMT2A
SCHEMBL530424 0.73 ALDH1A1 (0.51) ALDH1A1TSHRHTTKMT2ASMN1; SMN2
SCHEMBL7307357 0.71 ALDH1A1 (0.42) ALDH1A1TSHRHTTMAPK1KMT2A
SCHEMBL28706287 0.71 ALDH1A1 (0.42) ALDH1A1TSHRHTTMAPK1KMT2A
SCHEMBL11779225 0.71 ALDH1A1 (0.50) ALDH1A1TSHRHTTKMT2ASMN1; SMN2
SCHEMBL11091632 0.70 CES1 (0.53) ALDH1A1TSHRHTTKMT2ASMN1; SMN2
SCHEMBL3999764 0.70 ALDH1A1 (0.67) ALDH1A1TSHRHTTKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4675400-A FORM CONJUGATES WITH IMMUNOGLOBULINS; ANTITUMOR AGENTS ELI LILLY AND COMPANY (US) 1987-06-23 US claimed
EP-0153151-B1 TRANSFERRIN-VINCA ALKALOID CYTOTOXIC COMPOSITIONS ELI LILLY AND COMPANY (US) 1989-05-31 EP disclosed
EP-0153151-A2 Transferrin-vinca alkaloid cytotoxic compositions ELI LILLY AND COMPANY (US) 1985-08-28 EP disclosed
US-4522750-A Cytotoxic compositions of transferrin coupled to vinca alkaloids ELI LILLY AND COMPANY (US) 1985-06-11 US disclosed