SCHEMBL10608804

SCHEMBL10608804

CCCCC([O])c1ccc([N+](=O)[O-])c([N+](=O)[O-])c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.43
TSHR P16473 1/20 0.43
VCAM1 P19320 3/20 0.38
MAPT P10636 6/20 0.38
ALDH1A1 P00352 5/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
RXFP1 Q9HBX9 1/20 0.37
CASP6 P55212 1/20 0.37
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
STAT6 P42226 1/20 0.36
HIF1A Q16665 1/20 0.36
PHLPP2 Q6ZVD8 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HCAR3 P49019 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10611061 0.95 CYP3A4 (0.42) CYP3A4TSHRVCAM1MAPTALDH1A1
SCHEMBL10606953 0.94 CYP3A4 (0.41) CYP3A4TSHRVCAM1MAPTALDH1A1
SCHEMBL10608727 0.90 CYP3A4 (0.46) CYP3A4TSHRMAPTALDH1A1RXFP1
SCHEMBL10608523 0.83 CYP3A4 (0.48) CYP3A4TSHRMAPTALDH1A1TDP1
SCHEMBL10608761 0.79 MAPT (0.49) CYP3A4TSHRMAPTALDH1A1TDP1
SCHEMBL10608130 0.74 TSHR (0.59) CYP3A4TSHRVCAM1MAPTALDH1A1
SCHEMBL10607510 0.74 MAPT (0.47) CYP3A4TSHRMAPTALDH1A1TDP1
SCHEMBL9026356 0.73 ALDH1A1 (0.41) CYP3A4TSHRMAPTALDH1A1TDP1
SCHEMBL10607585 0.73 ASAH2 (0.47) CYP3A4TSHRMAPTALDH1A1TDP1
SCHEMBL10610870 0.73 ASAH2 (0.47) CYP3A4TSHRMAPTALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0162208-B1 NOVEL N-SUBSTITUTED 3,4-DIHYDROPYRIMIDINE DERIVATIVES, PROCESSES FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS SUNTORY KABUSHIKI KAISHA, also known as SUNTORY LTD. (JP) 1989-11-23 EP disclosed
US-4683234-A HYPOTENSIVE AGENTS, ANTI-ANGINA SUNTORY LIMITED (JP) 1987-07-28 US disclosed
EP-0162208-A2 Novel N-substituted 3,4-dihydropyrimidine derivatives, processes for preparing them and pharmaceutical compositions SUNTORY KABUSHIKI KAISHA, also known as SUNTORY LTD. (JP) 1985-11-27 EP disclosed