SCHEMBL10620665

SCHEMBL10620665

FC(F)(F)NCC1CCN(Cc2ccccc2)C1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.54
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
HIF1A Q16665 1/20 0.53
CCR3 P51677 1/20 0.53
DRD2 P14416 1/20 0.51
DRD4 P21917 1/20 0.51
DRD3 P35462 1/20 0.51
ACHE P22303 5/20 0.50
BCHE P06276 4/20 0.50
BACE1 P56817 4/20 0.50
KDM1A O60341 1/20 0.47
MAOB P27338 1/20 0.47
ALDH1A1 P00352 1/20 0.47
SLC6A4 P31645 1/20 0.46
SLC6A3 Q01959 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9688622 0.83 CXCR4 (0.58) CXCR4CYP1A2CYP2D6HIF1ACCR3
SCHEMBL28657725 0.81 CCR3 (0.57) CXCR4CYP1A2CYP2D6CCR3ACHE
SCHEMBL4923829 0.81 CXCR4 (0.61) CXCR4CYP1A2CYP2D6HIF1ACCR3
SCHEMBL11909092 0.80 HDAC3 (0.54) CXCR4DRD2DRD4DRD3ACHE
SCHEMBL5823 0.80 HDAC3 (0.54) CXCR4DRD2DRD4DRD3ACHE
SCHEMBL9437321 0.79 ACHE (0.60) CXCR4CYP1A2CYP2D6HIF1ACCR3
SCHEMBL10693231 0.79 CXCR4 (0.59) CXCR4CYP1A2CYP2D6HIF1ACCR3
SCHEMBL28788675 0.79 CCR3 (0.62) CXCR4CYP1A2CYP2D6HIF1ACCR3
SCHEMBL3810288 0.78 CXCR4 (0.62) CXCR4CYP1A2CYP2D6HIF1ACCR3
Hydrochloric Acid SCHEMBL10692701 0.78 CXCR4 (0.58) CXCR4CYP1A2CYP2D6HIF1ACCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4777175-A (NAPHTHYRIDINE, QUINOLINE) CARBOXYLIC ACID WARNER-LAMBERT COMPANY (US) 1988-10-11 US disclosed
US-4771054-A QUINOLINE CARBOXYLIC ACID WARNER-LAMBERT COMPANY (US) 1988-09-13 US disclosed
EP-0106489-B1 ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1988-07-27 EP disclosed
US-4665079-A QUINOLINE DERIVATIVES WARNER-LAMBERT COMPANY (US) 1987-05-12 US disclosed
US-4638067-A NAPHTHYRIDINE AND QUINOLINE CARBOXYLIC ACIDS WARNER-LAMBERT CO. (US) 1987-01-20 US disclosed
EP-0153163-A2 7-Substituted-1-cyclopropyl-6,8-difluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids; 7-substituted-1-cyclopropyl-1,4-dihydro-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acids; their derivatives; and a process for preparing the compounds WARNER-LAMBERT COMPANY (US) 1985-08-28 EP disclosed
EP-0106489-A2 Antibacterial agents WARNER-LAMBERT COMPANY (US) 1984-04-25 EP disclosed