SCHEMBL106285

SCHEMBL106285

CCn1nc(C)cc1C(=O)OC

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.52
GAA P10253 2/20 0.49
RAB9A P51151 1/20 0.49
ALDH1A1 P00352 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
LMNA P02545 2/20 0.45
KDM4E B2RXH2 2/20 0.45
POLB P06746 1/20 0.44
SMYD3 Q9H7B4 1/20 0.43
STING1 Q86WV6 5/20 0.42
PKM P14618 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
TBK1 Q9UHD2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6188814 0.86 MAPT (0.52) MAPTRAB9AALDH1A1NPSR1LMNA
SCHEMBL28556390 0.83 GAA (0.47) MAPTGAARAB9AALDH1A1LMNA
SCHEMBL23115927 0.83 AURKA (0.39) MAPTGAARAB9AALDH1A1NPSR1
SCHEMBL5108674 0.83 KDM4E (0.38) MAPTGAARAB9AALDH1A1NPSR1
SCHEMBL22857792 0.82 GAA (0.46) MAPTGAARAB9AALDH1A1NPSR1
SCHEMBL30514592 0.82 MAPT (0.49) MAPTALDH1A1NPSR1LMNAPOLB
SCHEMBL12688453 0.82 GAA (0.46) MAPTGAARAB9AALDH1A1NPSR1
SCHEMBL3817969 0.81 CA12 (0.37) MAPTGAARAB9AALDH1A1KDM4E
SCHEMBL31094892 0.81 KDM4E (0.38) MAPTGAARAB9AALDH1A1NPSR1
SCHEMBL23115866 0.81 CA12 (0.37) MAPTGAARAB9AALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12595249-B2 Aryl ether-substituted heterocyclic compounds as glpir agonists MINDRANK AI LTD. (CN) 2026-04-07 US disclosed
US-12497384-B2 Aryl ether-substituted heterocyclic compounds as GLP1R agonists MINDRANK AI LTD. (CN) 2025-12-16 US disclosed
US-20250304553-A1 ARYL ETHER-SUBSTITUTED HETEROCYCLIC COMPOUNDS AS GLP1R AGONISTS MINDRANK AI LTD. (CN) 2025-10-02 US disclosed
US-20250282757-A1 ARYL ETHER-SUBSTITUTED HETEROCYCLIC COMPOUNDS AS GLP1R AGONISTS MINDRANK AI LTD. (CN) 2025-09-11 US disclosed
EP-4526298-A1 PYRAZOLE DERIVATIVES AS STING AGONISTS F. Hoffmann-La Roche AG (CH) 2025-03-26 EP disclosed
CN-117242067-B Novel aryl ether substituted heterocycles as GLP1R agonists 杭州德睿智药科技有限公司 2025-03-25 CN disclosed
US-20250074913-A1 PYRAZOLE DERIVATIVES AS STING AGONISTS HOFFMANN-LA ROCHE INC. (US) 2025-03-06 US disclosed
CN-119212989-A Pyrazole derivatives as STING agonists 豪夫迈·罗氏有限公司 2024-12-27 CN disclosed
EP-4353717-A1 NOVEL ARYL ETHER SUBSTITUTED HETEROCYCLIC COMPOUND AS GLP1R AGONIST Mindrank AI Ltd. (CN) 2024-04-17 EP disclosed
WO-2024051700-A1 NOVEL ARYL DEUTERATED BENZYL ETHER SUBSTITUTED HETEROCYCLIC COMPOUND AS GLP1R AGONIST 德睿智药(苏州)新药研发有限公司 2024-03-14 WO disclosed
US-8455532-B2 Pyrazolyl acrylonitrile compounds and uses thereof SHENYANG RESEARCH INSTITUTE OF CHEMICAL INDUSTRY CO., LTD. (CN) 2013-06-04 US disclosed
US-8455532-B2 Pyrazolyl acrylonitrile compounds and uses thereof SHENYANG RESEARCH INSTITUTE OF CHEMICAL INDUSTRY CO., LTD. (CN) 2013-06-04 US disclosed
US-8455532-B2 Pyrazolyl acrylonitrile compounds and uses thereof SHENYANG RESEARCH INSTITUTE OF CHEMICAL INDUSTRY CO., LTD. (CN) 2013-06-04 US disclosed
EP-2426110-A1 PYRAZOLYL ACRYLONITRILE COMPOUNDS AND USES THEREOF Sinochem Corporation (CN) 2012-03-07 EP disclosed
EP-2426110-A1 PYRAZOLYL ACRYLONITRILE COMPOUNDS AND USES THEREOF Sinochem Corporation (CN) 2012-03-07 EP disclosed
US-20120035236-A1 Pyrazolyl Acrylonitrile Compounds and Uses Thereof SHENYANG SINOCHEM AGROCHEMICALS R&D CO., LTD. (CN) 2012-02-09 US disclosed
US-20120035236-A1 Pyrazolyl Acrylonitrile Compounds and Uses Thereof SHENYANG SINOCHEM AGROCHEMICALS R&D CO., LTD. (CN) 2012-02-09 US disclosed
US-20120035236-A1 Pyrazolyl Acrylonitrile Compounds and Uses Thereof SHENYANG SINOCHEM AGROCHEMICALS R&D CO., LTD. (CN) 2012-02-09 US disclosed
EP-0087780-B2 Pyrazolesulfonylurea derivative, preparation thereof, herbicide containing said derivative as active ingredient and herbicidal method by use thereof NISSAN CHEMICAL IND LTD (JP) 1995-02-15 EP disclosed
US-4954164-A Pyrazolesulfonylurea derivatives, preparation thereof, herbicide containing said derivative as active ingredient and herbicidal method by use thereof NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 1990-09-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12497384-B2 Aryl ether-substituted heterocyclic compounds as GLP1R agonists GLP1R, GIPR, GCGR MAPT 3780/4885GAA 2562/4885RAB9A 592/4885
US-12595249-B2 Aryl ether-substituted heterocyclic compounds as glpir agonists GLP1R, GIPR, GCGR MAPT 4801/4885GAA 4195/4885RAB9A 1015/4885
US-20250304553-A1 ARYL ETHER-SUBSTITUTED HETEROCYCLIC COMPOUNDS AS GLP1R AGONISTS GLP1R, GIPR, GCGR MAPT 3889/4885GAA 2003/4885RAB9A 827/4885
US-20250074913-A1 PYRAZOLE DERIVATIVES AS STING AGONISTS STING1, CGAS, MAVS MAPT 4128/4885GAA 3157/4885RAB9A 413/4885
US-20250282757-A1 ARYL ETHER-SUBSTITUTED HETEROCYCLIC COMPOUNDS AS GLP1R AGONISTS GLP1R, GIPR, GCGR MAPT 3591/4885GAA 2478/4885RAB9A 563/4885
US-20120035236-A1 Pyrazolyl Acrylonitrile Compounds and Uses Thereof CBR3, C3AR1, C5 MAPT 4805/4885GAA 4389/4885RAB9A 2342/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.