SCHEMBL10638080

SCHEMBL10638080

COc1ccc(C(=O)C2CCN(C(=O)O)CC2)c(O)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CPS1 P31327 1/20 0.60
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
POLB P06746 1/20 0.51
HSD11B1 P28845 3/20 0.51
ALDH1A1 P00352 6/20 0.50
HPGD P15428 3/20 0.50
MAPK1 P28482 2/20 0.50
CYP3A4 P08684 2/20 0.50
LMNA P02545 5/20 0.48
HTT P42858 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
GAA P10253 1/20 0.48
CYP1A2 P05177 2/20 0.48
PGR P06401 2/20 0.48
SLC6A2 P23975 2/20 0.48
CYP2C19 P33261 2/20 0.48
CYP2D6 P10635 1/20 0.48
PDE4A P27815 1/20 0.48
HRH1 P35367 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10634871 0.90 CPS1 (0.60) CPS1NPC1RAB9APOLBHSD11B1
SCHEMBL10637442 0.81 MEN1 (0.57) ALDH1A1
SCHEMBL10637499 0.81 NPC1 (0.57) CPS1NPC1RAB9AALDH1A1HPGD
Hydrochloric Acid SCHEMBL10640839 0.80 NPC1 (0.55) CPS1NPC1RAB9AALDH1A1HPGD
SCHEMBL10637691 0.80 CPS1 (0.47) CPS1NPC1RAB9AHSD11B1ALDH1A1
SCHEMBL10638084 0.80 CPS1 (0.47) CPS1NPC1RAB9AHSD11B1ALDH1A1
SCHEMBL4962237 0.79 POLB (0.78) NPC1RAB9APOLBHSD11B1ALDH1A1
SCHEMBL10638070 0.79 CPS1 (0.57) CPS1POLBHSD11B1ALDH1A1LMNA
SCHEMBL14638260 0.78 MGLL (0.66) POLBHSD11B1ALDH1A1LMNAMGLL
SCHEMBL11195650 0.77 CPS1 (0.45) CPS1NPC1RAB9AHSD11B1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4408053-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1983-10-04 US claimed
EP-0080104-B1 3-(4-PIPERIDYL)-1,2-BENZISOXAZOLES, PROCESS FOR THE PREPARATION THEREOF, AND A PHARMACEUTICAL COMPOSITION COMPRISING THE SAME HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1988-12-14 EP disclosed
US-4528376-A 3-(4-Piperidyl)-1,2-benzisoxazoles HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1985-07-09 US disclosed
US-4469869-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1984-09-04 US disclosed
US-4408053-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1983-10-04 US disclosed
US-4408054-A ANALGESTICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1983-10-04 US disclosed
EP-0080104-A2 3-(4-Piperidyl)-1,2-benzisoxazoles, process for the preparation thereof, and a pharmaceutical composition comprising the same HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1983-06-01 EP disclosed
US-4355037-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS (US) 1982-10-19 US disclosed