SCHEMBL10646248

SCHEMBL10646248

c1csc(Cn2cnnc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.45
TSHR P16473 3/20 0.44
KDM4E B2RXH2 2/20 0.44
TAAR1 Q96RJ0 1/20 0.43
DRD4 P21917 7/20 0.43
DRD3 P35462 4/20 0.43
ALDH1A1 P00352 2/20 0.41
MAPT P10636 2/20 0.41
HSD17B10 Q99714 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HPGD P15428 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
DRD5 P21918 2/20 0.40
DRD2 P14416 2/20 0.40
CYP2C19 P33261 1/20 0.38
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL448303 0.80 HTT (0.50) HTTL3MBTL1TSHRKDM4ETAAR1
SCHEMBL9369294 0.79 CYP11B1 (0.55) MAPT
SCHEMBL8309874 0.75 HTT (0.42) HTTL3MBTL1TSHRKDM4ETAAR1
SCHEMBL3842559 0.74 ALDH1A1 (0.45) HTTL3MBTL1TSHRKDM4ETAAR1
SCHEMBL14204090 0.72 HTT (0.40) HTTL3MBTL1TSHRKDM4ETAAR1
SCHEMBL3120892 0.71 CYP19A1 (0.53) HTTL3MBTL1TSHRKDM4ETAAR1
SCHEMBL14833178 0.71 CYP19A1 (0.53) HTTL3MBTL1TSHRKDM4EDRD4
SCHEMBL4943132 0.70 KDM4E (0.49) HTTL3MBTL1TSHRKDM4EALDH1A1
SCHEMBL1037058 0.68 HTT (0.66) HTTTSHRKDM4EDRD4DRD3
SCHEMBL10648832 0.68 HTT (0.43) HTTL3MBTL1TSHRKDM4ETAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0128502-B1 SUBSTITUTED 6-(THIEN-2-YL)-3(2H)-PYRIDAZINONES AND PROCESSES FOR THEIR PREPARATION A. Nattermann & Cie. GmbH (DE) 1988-08-31 EP disclosed
EP-0128502-A1 Substituted 6-(thien-2-yl)-3(2H)-pyridazinones and processes for their preparation A. Nattermann & Cie. GmbH (DE) 1984-12-19 EP disclosed