SCHEMBL10646593

SCHEMBL10646593

CCOc1cc2cc(C(=O)O)sc2cc1O

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 1/20 0.61
STING1 Q86WV6 14/20 0.51
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
BCL2L1 Q07817 1/20 0.41
CLK1 P49759 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tibenelast SCHEMBL449748 0.89 STING1 (0.54) GPR35STING1ALDH1A1HPGDTDP1
SCHEMBL10645446 0.89 STING1 (0.49) GPR35STING1CLK1HDAC3HDAC4
Tibenelast SCHEMBL10688452 0.88 STING1 (0.53) GPR35STING1ALDH1A1HPGDTDP1
Tibenelast SCHEMBL635433 0.88 STING1 (0.53) GPR35STING1ALDH1A1HPGDTDP1
SCHEMBL10641965 0.84 STING1 (0.60) STING1
SCHEMBL10642176 0.84 STING1 (0.60) STING1
SCHEMBL1608203 0.83 GPR35 (0.67) GPR35STING1HDAC3HDAC4HDAC1
SCHEMBL10537567 0.83 STING1 (0.49) GPR35STING1ALDH1A1HPGDTDP1
SCHEMBL10534791 0.83 STING1 (0.49) GPR35STING1ALDH1A1HPGDTDP1
SCHEMBL10642801 0.82 STING1 (0.56) GPR35STING1ALDH1A1HPGDTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0139464-B1 BENZOTHIOPHENE DERIVATES AS BRONCHODILATORS ELI LILLY AND COMPANY (US) 1988-10-19 EP disclosed
US-4552891-A BRONCHODILATOR ELI LILLY AND COMPANY (US) 1985-11-12 US disclosed
EP-0139464-A1 Benzothiophene derivates as bronchodilators ELI LILLY AND COMPANY (US) 1985-05-02 EP disclosed