SCHEMBL10651209

SCHEMBL10651209

COc1cc(CCC(C)N)cc(NS(C)(=O)=O)c1OC

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.49
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA9 Q16790 2/20 0.49
CA14 Q9ULX7 2/20 0.49
HTR2A P28223 2/20 0.41
HTR2C P28335 2/20 0.41
HTR2B P41595 2/20 0.41
ADRB3 P13945 6/20 0.40
CYP19A1 P11511 1/20 0.38
AOC3 Q16853 1/20 0.38
G6PD P11413 1/20 0.37
LMNA P02545 1/20 0.37
CA5A P35218 1/20 0.36
PTK2 Q05397 3/20 0.36
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10753256 0.78 CA12 (0.47) CA12CA1CA2CA9CA14
SCHEMBL26673643 0.70 PTK2 (0.42) CA12CA1CA2CA9CA14
SCHEMBL690776 0.69 ADRB3 (0.37) CA12CA1CA2CA9CA14
SCHEMBL9253296 0.67 HTR2A (0.60) CA12CA1CA2CA9CA14
SCHEMBL10651132 0.67 KDM4E (0.58) CA12CA1CA2CA9ADRB3
SCHEMBL27673619 0.67 HTR2A (0.59) CA12CA1CA2CA9CA14
SCHEMBL265633 0.67 STAT3 (0.63) CA12CA1CA2CA9CA14
SCHEMBL10652433 0.66 NR3C1 (0.48)
SCHEMBL5673172 0.66 KDM4E (0.57) CA12CA1CA2CA9CA14
SCHEMBL689520 0.66 ADRB3 (0.38) ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0157267-B1 SUBSTITUTED BENZOPYRANS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN MEDICINES BAYER AG (DE) 1988-11-23 EP disclosed
US-4659737-A Substituted aminomethyl benzopyrans having anti-hypertensive activities BAYER AKTIENGESELLSCHAFT (DE) 1987-04-21 US disclosed
US-4647579-A Circulation active novel substituted 4-hydroxy-benzopyrans BAYER AKTIENGESELLSCHAFT (DE) 1987-03-03 US disclosed
EP-0158164-A2 Substituted 4-hydroxy-benzopyrans, process for their preparation and their use in medicines BAYER AG (DE) 1985-10-16 EP disclosed
EP-0157267-A2 Substituted benzopyrans, process for their preparation and their use in medicines BAYER AG (DE) 1985-10-09 EP disclosed