SCHEMBL10651972

SCHEMBL10651972

CCc1nc(N)nc(N)c1N1CCN(c2ccc(C(=O)N[C@@H](CCC(N)=O)C(=O)O)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DHFR P00374 13/20 0.54
MTR Q99707 1/20 0.53
TYMS P04818 2/20 0.47
CA2 P00918 2/20 0.45
CA1 P00915 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6699116 0.94 DHFR (0.61) DHFRMTRTYMS
SCHEMBL10647855 0.93 DHFR (0.56) DHFRMTRTYMSCA2CA1
SCHEMBL10652925 0.90 DHFR (0.58) DHFRMTRTYMSCA2CA1
SCHEMBL6701864 0.87 DHFR (0.59) DHFRMTRTYMS
SCHEMBL6697447 0.84 DHFR (0.54) DHFRMTR
SCHEMBL6704122 0.83 DHFR (0.66) DHFRMTRTYMS
SCHEMBL6701226 0.79 DHFR (0.73) DHFR
SCHEMBL6699847 0.78 DHFR (0.52) DHFRMTR
SCHEMBL6705312 0.76 DHFR (0.49) DHFRMTR
SCHEMBL11125686 0.73 DHFR (0.57) DHFRMTRTYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0103464-B1 DIAMINOPYRIMIDINES AND THEIR PRODUCTION WARNER-LAMBERT COMPANY (US) 1988-11-17 EP claimed