SCHEMBL10653154

SCHEMBL10653154

CCOC(=O)CC(CO)CC(C)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGAM O43451 1/20 0.43
GAA P10253 1/20 0.43
SI P14410 1/20 0.43
MGAM2 Q2M2H8 1/20 0.43
ALDH1A1 P00352 8/20 0.40
TRPA1 O75762 1/20 0.40
HSD17B10 Q99714 2/20 0.39
LMNA P02545 1/20 0.39
ALOX15 P16050 3/20 0.38
CYP3A4 P08684 2/20 0.38
TSHR P16473 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
CHRM1 P11229 1/20 0.37
ADORA1 P30542 1/20 0.37
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HTT P42858 1/20 0.33
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5000280 0.87 MGAM (0.50) MGAMGAASIMGAM2ALDH1A1
SCHEMBL10405753 0.83 MGAM (0.46) MGAMGAASIMGAM2ALDH1A1
SCHEMBL15187255 0.80 MGAM (0.43) MGAMGAASIMGAM2ALDH1A1
SCHEMBL15187221 0.80 MGAM (0.43) MGAMGAASIMGAM2ALDH1A1
SCHEMBL28262928 0.80 MGAM (0.43) MGAMGAASIMGAM2ALDH1A1
SCHEMBL14513819 0.80 ALDH1A1 (0.50) ALDH1A1TRPA1LMNATSHRTDP1
SCHEMBL8057583 0.78 MGAM (0.41) MGAMGAASIMGAM2ALDH1A1
SCHEMBL15187368 0.77 ALDH1A1 (0.50) MGAMGAASIMGAM2ALDH1A1
SCHEMBL234553 0.76 MGAM (0.52) MGAMGAASIMGAM2ALDH1A1
SCHEMBL1456370 0.76 MGAM (0.52) MGAMGAASIMGAM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4751246-A ALPHA(AMINOALKYL)-4-HYDROXY-3-(ALKYLSULFINYL) BENZENEMETHANOL AND 2-(4-HYDROXY-3-(ALKYLSULFINYL) PHENYL)ETHYLAMINE-HYPOTENSIVE AGENTS STERLING DRUG INC. (US) 1988-06-14 US disclosed
US-4452816-A HYPOTENSIVE AND ANTIARRHYTHMIA AGENTS STERLING DRUG INC. (US) 1984-06-05 US disclosed
US-4374149-A HYPOTENSIVE AGENT AND VASODILATOR STERLING DRUG INC. (US) 1983-02-15 US disclosed
US-4255564-A ANTIBIOTICS, PROTECTED ALDEHYDE GROUP, INTERMEDIATES ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1981-03-10 US disclosed
US-4196280-A Novel macrolactone derivatives and process of producing them ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1980-04-01 US disclosed