SCHEMBL10653335

SCHEMBL10653335

COc1nc2ccccc2c(OC)c1-c1ccccc1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.54
ADORA2A P29274 2/20 0.44
CYP1A2 P05177 5/20 0.42
CYP2D6 P10635 3/20 0.42
CLK4 Q9HAZ1 3/20 0.42
CYP3A4 P08684 3/20 0.42
MAPK1 P28482 3/20 0.42
CYP2C19 P33261 2/20 0.42
HSD17B10 Q99714 2/20 0.42
TSHR P16473 2/20 0.42
USP2 O75604 1/20 0.42
ALOX15 P16050 1/20 0.42
LMNA P02545 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KDM4E B2RXH2 2/20 0.41
ADORA3 P0DMS8 1/20 0.40
MAPT P10636 2/20 0.39
BACE1 P56817 1/20 0.39
MEN1 O00255 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4272933 0.77 POLB (0.66) POLBCYP1A2CYP3A4MAPK1CYP2C19
SCHEMBL29450270 0.77 POLB (0.70) POLBCYP1A2CYP3A4MAPK1CYP2C19
SCHEMBL9694998 0.77 POLB (0.70) POLBCYP1A2CYP3A4MAPK1CYP2C19
SCHEMBL19608972 0.75 ADORA2A (0.56) POLBADORA2ACYP1A2CYP2D6CLK4
SCHEMBL3731388 0.74 ALDH1A1 (0.50) POLBADORA2ACYP1A2CYP2D6CLK4
Hydrochloric Acid SCHEMBL10648998 0.73 TOP2A (0.52)
SCHEMBL31061121 0.72 CYP1A2 (0.63) POLBADORA2ACYP1A2CYP2D6CLK4
SCHEMBL23145043 0.72 POLB (0.63) POLBADORA2ACYP1A2CYP3A4MAPK1
SCHEMBL1408391 0.72 POLB (1.00) POLBMAPK1HSD17B10TSHRLMNA
SCHEMBL5457232 0.72 ALDH1A1 (0.44) POLBADORA2ACYP1A2MAPK1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0093521-B1 QUINOLINE DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-08-24 EP disclosed
US-4607039-A 2-(AMINO-ALKYL-THIO OR -OXY) SUBSTITUTED IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-08-19 US disclosed
EP-0093521-A2 Quinoline derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1983-11-09 EP disclosed