SCHEMBL10653784

SCHEMBL10653784

CN(CCCN)c1ccc(Br)cn1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 6/20 0.57
HRH3 Q9Y5N1 2/20 0.50
RAD52 P43351 1/20 0.41
SSTR2 P30874 4/20 0.39
SSTR4 P31391 4/20 0.39
HCAR3 P49019 1/20 0.39
PKM P14618 1/20 0.34
AOC3 Q16853 1/20 0.34
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
EGFR P00533 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5237488 0.86 GBA1 (0.60) GBA1HRH3SSTR2SSTR4HCAR3
SCHEMBL2256335 0.85 GBA1 (0.51) GBA1HRH3SSTR2SSTR4HCAR3
SCHEMBL31217157 0.85 GBA1 (0.56) GBA1HCAR3AOC3NPC1RAB9A
SCHEMBL9866571 0.81 HRH3 (0.51) GBA1HRH3HCAR3PKMAOC3
SCHEMBL1432671 0.81 GBA1 (0.59) GBA1HCAR3PKMAOC3NPC1
SCHEMBL21841697 0.81 GBA1 (0.47) GBA1RAD52SSTR2SSTR4HCAR3
SCHEMBL5255404 0.79 GBA1 (0.53) GBA1SSTR2SSTR4HCAR3NPC1
SCHEMBL1433090 0.77 GBA1 (0.69) GBA1HCAR3AOC3NPC1ALDH1A1
SCHEMBL5253357 0.77 GBA1 (0.50) GBA1HCAR3ALDH1A1EGFR
SCHEMBL14484960 0.76 HRH3 (0.47) GBA1HRH3HCAR3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0113572-B1 PYRIDINE DERIVATIVES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1988-02-03 EP disclosed
US-4547506-A 2-Pyridylaminoakylamino-4-pyrimidones useful as histamine H1 -antagonists SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1985-10-15 US disclosed
EP-0113572-A2 Pyridine derivatives SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1984-07-18 EP disclosed