SCHEMBL10657017

SCHEMBL10657017

CC(C)(C)OC(=O)NC(Cc1ccc(O)c(C(C)(C)C)c1)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.57
ITGB3 P05106 2/20 0.54
ITGA2B P08514 2/20 0.54
PTPN1 P18031 1/20 0.52
CTSS P25774 8/20 0.51
CTSK P43235 7/20 0.51
CTSB P07858 3/20 0.49
PPARA Q07869 5/20 0.49
PPARG P37231 4/20 0.49
ITGB1 P05556 1/20 0.48
ITGAV P06756 1/20 0.48
ITGB5 P18084 1/20 0.48
PPARD Q03181 2/20 0.47
CTSL P07711 1/20 0.47
ITGA4 P13612 1/20 0.47
ITGB7 P26010 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10657027 1.00 ACE (0.57) ACEITGB3ITGA2BPTPN1CTSS
SCHEMBL23447587 0.89 KLK5 (0.52) ACECTSSCTSKCTSBCTSL
SCHEMBL4786137 0.89 ACE (0.60) ACEITGB3ITGA2BPTPN1CTSS
SCHEMBL1172086 0.89 ACE (0.60) ACEITGB3ITGA2BPTPN1CTSS
SCHEMBL30829409 0.89 ACE (0.60) ACEITGB3ITGA2BPTPN1CTSS
SCHEMBL31525018 0.88 ACE (0.59) ACEITGB3ITGA2BPTPN1CTSS
SCHEMBL15565481 0.86 ACE (0.58) ACEITGB3ITGA2BPTPN1CTSS
SCHEMBL13286814 0.86 ACE (0.58) ACEITGB3ITGA2BPTPN1CTSS
SCHEMBL24489644 0.85 FOLH1 (0.62) ACEITGB3ITGA2BPTPN1CTSS
SCHEMBL2631434 0.85 PTPN1 (0.59) ACEITGB3ITGA2BPTPN1CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4722922-A RENIN INHIBITION G. D. SEARLE & CO. (US) 1988-02-02 US disclosed
US-4603121-A ANALGESICS G. D. SEARLE & CO. (US) 1986-07-29 US disclosed
EP-0136720-A2 Enkephalin analogs G.D. Searle & Co. (US) 1985-04-10 EP disclosed
US-4495178-A Enkephalin analogs G. D. SEARLE & CO. (US) 1985-01-22 US disclosed