SCHEMBL10658249

SCHEMBL10658249

COc1cc2c(cc1O)CCN(CCc1ccc(N)cc1)C2C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.57
DRD2 P14416 2/20 0.51
DRD1 P21728 2/20 0.51
DRD3 P35462 1/20 0.51
SIGMAR1 Q99720 1/20 0.51
TBXA2R P21731 1/20 0.51
DHCR7 Q9UBM7 2/20 0.49
TP53 P04637 1/20 0.48
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
GAA P10253 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
KCNH2 Q12809 1/20 0.46
BCHE P06276 1/20 0.45
ACHE P22303 1/20 0.45
ABCB1 P08183 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
DHFR P00374 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10662154 0.99 MAOA (0.59) MAOADRD2DRD1DRD3SIGMAR1
Veradoline SCHEMBL29388371 0.91 MAOA (0.53) MAOAMAPK1KDM4EALDH1A1ABCB1
Veradoline SCHEMBL489286 0.91 MAOA (0.53) MAOAMAPK1KDM4EALDH1A1ABCB1
Veradoline SCHEMBL10656736 0.90 MAOA (0.55) MAOAMAPK1KDM4EALDH1A1ABCB1
Veradoline SCHEMBL125027 0.90 MAOA (0.55) MAOAMAPK1KDM4EALDH1A1ABCB1
SCHEMBL10659587 0.89 MAOA (0.52) MAOADRD2DRD1DRD3SIGMAR1
Bromide SCHEMBL10656534 0.88 MAOA (0.51) MAOADRD2DRD1DRD3SIGMAR1
SCHEMBL10662687 0.84 KDM4E (0.61) MAOADRD2DRD1DRD3SIGMAR1
Hydrochloric Acid SCHEMBL10662226 0.83 KDM4E (0.60) MAOADRD2DRD1DRD3SIGMAR1
SCHEMBL10659360 0.81 CA1 (0.49) DRD2DRD1DRD3SIGMAR1ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4766131-A 2-amino (or hydroxy) phenethyl-1,2,3,4-tetrahydroisoquinolines as analgesics PENNWALT CORPORATION (US) 1988-08-23 US claimed
EP-0051190-A2 N-(amino(or hydroxy) phenethyl)-1,2,3,4-tetrahydroisoquinolines, precursors thereof, and methods of preparation PENNWALT CORPORATION (US) 1982-05-12 EP claimed