SCHEMBL10667192

SCHEMBL10667192

COc1cc2c(cc1OC)CC(=O)N(CCCN(C)CCc1coc3ccccc13)C=C2

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCN4 Q9Y3Q4 6/20 0.48
BRD4 O60885 1/20 0.43
SMPD1 P17405 4/20 0.42
MAPT P10636 1/20 0.41
CYP3A4 P08684 1/20 0.40
ALOX15 P16050 1/20 0.40
ABCB1 P08183 1/20 0.36
PDE10A Q9Y233 1/20 0.35
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
MAOA P21397 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10666609 0.90 HCN4 (0.47) HCN4BRD4SMPD1MAPTCYP3A4
SCHEMBL10894643 0.83 HCN4 (0.48) HCN4BRD4SMPD1MAPTCYP3A4
SCHEMBL10669932 0.83 HCN4 (0.50) HCN4BRD4SMPD1MAPTCYP3A4
Hydrochloric Acid SCHEMBL10667216 0.82 HCN4 (0.49) HCN4BRD4SMPD1MAPTCYP3A4
SCHEMBL10664298 0.82 HCN4 (0.49) HCN4BRD4SMPD1MAPTCYP3A4
SCHEMBL10664291 0.82 HCN4 (0.38) HCN4SMPD1MAPT
SCHEMBL10670888 0.81 HCN4 (0.51) HCN4BRD4SMPD1MAPTCYP3A4
SCHEMBL10663997 0.81 HCN4 (0.64) HCN4SMPD1MAPTCYP3A4ALOX15
Hydrochloric Acid SCHEMBL10671903 0.81 HCN4 (0.51) HCN4BRD4SMPD1MAPTCYP3A4
SCHEMBL10663974 0.80 MAPT (0.40) HCN4SMPD1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4737495-A ANTIALLERGENS, ANTISCHEMIC, HYPOTENSIVE AGENTS DR. KARL TOMAE, GMBH (DE) 1988-04-12 US disclosed
EP-0204349-A2 Heteroaromatic amine derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1986-12-10 EP disclosed