SCHEMBL10668147

SCHEMBL10668147

O=C(CNC(=O)c1ccccc1)N[C@@H](CS)C(=O)N1CCC[C@H]1C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.56
ACE P12821 14/20 0.53
ACE2 Q9BYF1 8/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9509731 0.82 ACE (0.66) TSHRACEACE2
SCHEMBL9551626 0.82 ACE (0.66) TSHRACEACE2
SCHEMBL10668559 0.81 ACE (0.68) TSHRACEACE2
SCHEMBL22811348 0.79 PREP (0.69) ACEACE2
SCHEMBL22209470 0.79 PREP (0.69) ACEACE2
SCHEMBL9509127 0.78 ACE (0.63) TSHRACEACE2
SCHEMBL30905695 0.77 ACE (0.48) ACEACE2
SCHEMBL10830758 0.77 TSHR (0.62) TSHRACEACE2
SCHEMBL10830200 0.77 TSHR (0.62) TSHRACEACE2
SCHEMBL15251975 0.77 ACE (0.70) TSHRACEACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4745124-A THIO/ESTER PEPTIDES UNIVERSITY OF MIAMI (US) 1988-05-17 US disclosed
US-4695582-A Inhibitors of angiotensin converting enzyme UNIVERSITY OF MIAMI (US) 1987-09-22 US disclosed