SCHEMBL10678652

SCHEMBL10678652

Cc1ccc(S(=O)(=O)OCC2CCc3cc(Br)ccc3C2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.42
ALDH1A1 P00352 3/20 0.42
CYP3A4 P08684 2/20 0.42
TSHR P16473 2/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42
SGPL1 O95470 3/20 0.37
S1PR1 P21453 3/20 0.37
MCHR1 Q99705 3/20 0.37
CYP26A1 O43174 1/20 0.36
CYP19A1 P11511 1/20 0.36
CYP11B2 P19099 1/20 0.35
ADRA2A P08913 1/20 0.35
PNMT P11086 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
DPP4 P27487 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7296513 0.85 CYP19A1 (0.52) CYP26A1CYP19A1
SCHEMBL7380518 0.83 CYP19A1 (0.41) ALDH1A1SGPL1S1PR1MCHR1CYP19A1
SCHEMBL7719725 0.83 PSEN1 (0.46) CYP2D6ALDH1A1TSHRS1PR1CYP19A1
SCHEMBL6197173 0.81 MCHR1 (0.45) ALDH1A1TSHRCYP2C9MAPTMAPK1
SCHEMBL9630809 0.81 CYP19A1 (0.52) CYP26A1CYP19A1
SCHEMBL10529517 0.80 GAA (0.46) ALDH1A1TSHRCYP2C9MAPTMAPK1
SCHEMBL7723979 0.77 PSEN1 (0.47) CYP2D6ALDH1A1CYP3A4CYP2C19MAPK1
SCHEMBL31267611 0.77 CYP2D6 (0.41) CYP2D6ALDH1A1CYP3A4TSHRCYP2C9
SCHEMBL4225647 0.76 CYP19A1 (0.47) ALDH1A1CYP26A1CYP19A1
SCHEMBL10532540 0.75 GAA (0.46) ALDH1A1TSHRCYP2C9MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4777257-A CARDIOVASCULAR DISORDERS DAIICHI SEIYAKU CO., LTD. (JP) 1988-10-11 US disclosed
US-4665188-A Certain [(1-imidazolyl)-lower-alkylene]-tetrahydronaphthalenecarboxylic acids or corresponding idan-carboxylic acids which are thromboxane A2 DAIICHI SEIYAKU CO., LTD. (JP) 1987-05-12 US disclosed
EP-0135177-A2 Benzocycloalkane derivatives DAIICHI SEIYAKU CO., LTD. (JP) 1985-03-27 EP disclosed