SCHEMBL9630809

SCHEMBL9630809

COc1ccc2c(c1)CC(COS(=O)(=O)c1ccc(C)cc1)CC2

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.52
DRD2 P14416 5/20 0.49
DRD3 P35462 5/20 0.49
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
ACHE P22303 2/20 0.46
CYP26A1 O43174 1/20 0.46
HTR1A P08908 2/20 0.46
SIGMAR1 Q99720 1/20 0.46
DRD4 P21917 2/20 0.45
MTNR1A P48039 1/20 0.45
MTNR1B P49286 1/20 0.45
HTR6 P50406 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7296513 0.95 CYP19A1 (0.52) CYP19A1DRD2DRD3CA1CA2
SCHEMBL4225647 0.91 CYP19A1 (0.47) CYP19A1DRD2DRD3CA1CA2
SCHEMBL7719725 0.83 PSEN1 (0.46) CYP19A1DRD2CA1CA2
SCHEMBL6401807 0.81 DRD2 (0.50) CYP19A1DRD2DRD3CA1CA2
SCHEMBL10678652 0.81 CYP2D6 (0.42) CYP19A1CYP26A1
SCHEMBL10532540 0.80 GAA (0.46) DRD2DRD3CA1CA2
SCHEMBL7776659 0.79 CHRM2 (0.58) CYP19A1DRD2DRD3CA1CA2
SCHEMBL7380518 0.79 CYP19A1 (0.41) CYP19A1ACHE
SCHEMBL6197173 0.78 MCHR1 (0.45)
SCHEMBL8765272 0.77 CYP2D6 (0.45) DRD2DRD3CA1CA2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0213080-B1 HYDROGENATED PYRIDINE DERIVATIVES CIBA-GEIGY AG (CH) 1992-05-20 EP disclosed
EP-0213080-A2 Hydrogenated pyridine derivatives CIBA-GEIGY AG (CH) 1987-03-04 EP disclosed