SCHEMBL10679403

SCHEMBL10679403

OC(CC1CCCCN1)c1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.62
POLB P06746 1/20 0.54
CACNA2D1 P54289 1/20 0.51
CACNA1B Q00975 1/20 0.51
CACNB1 Q02641 1/20 0.51
CYP1A2 P05177 1/20 0.50
HIF1A Q16665 1/20 0.50
SLC6A3 Q01959 6/20 0.49
SLC6A2 P23975 5/20 0.49
SLC6A4 P31645 4/20 0.49
DHFR P00374 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22259900 0.95 CYP2D6 (0.56) CYP2D6POLBCACNA2D1CACNA1BCACNB1
SCHEMBL20833013 0.95 CYP2D6 (0.56) CYP2D6POLBCACNA2D1CACNA1BCACNB1
SCHEMBL8507267 0.95 CYP2D6 (0.56) CYP2D6POLBCACNA2D1CACNA1BCACNB1
SCHEMBL20832991 0.95 CYP2D6 (0.56) CYP2D6POLBCACNA2D1CACNA1BCACNB1
SCHEMBL465920 0.89 CYP2D6 (0.58) CYP2D6POLBCACNA2D1CACNA1BCACNB1
SCHEMBL8493732 0.85 POLB (0.59) CYP2D6POLBCACNA2D1CACNA1BCACNB1
SCHEMBL5949168 0.84 CYP2D6 (0.56) CYP2D6POLBCACNA2D1CACNA1BCACNB1
SCHEMBL6560565 0.84 CYP2D6 (0.56) CYP2D6POLBCACNA2D1CACNA1BCACNB1
SCHEMBL6560568 0.84 CYP2D6 (0.56) CYP2D6POLBCACNA2D1CACNA1BCACNB1
SCHEMBL465909 0.84 CYP2D6 (0.53) CYP2D6POLBSLC6A3SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4780478-A Aminopropoxy-chromones useful as antidepressants MERCK PATENT GESELLSCHAFT MIT BERSCHRANKTER HAFTUNG (DE) 1988-10-25 US disclosed
US-4508732-A Basic ethers useful as antidepressant agents MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1985-04-02 US disclosed
EP-0031885-B1 BASIC ETHERS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR THEIR PREPARATION MERCK PATENT GmbH (DE) 1984-06-27 EP disclosed
US-4376123-A Hexahydroazepinyloxy-chromones useful as antidepressants MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1983-03-08 US disclosed
EP-0031885-A1 Basic ethers, pharmaceutical compositions containing them and process for their preparation MERCK PATENT GmbH (DE) 1981-07-15 EP disclosed
US-4225608-A ANTIDEPRESSANTS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1980-09-30 US disclosed