SCHEMBL10683407

SCHEMBL10683407

O=C(O)c1cn(C2CC2)c2cc(N3CCC(O)C3)c(F)c(F)c2c1=O

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.64
HRH3 Q9Y5N1 1/20 0.64
ALDH1A1 P00352 5/20 0.50
KDM4E B2RXH2 4/20 0.50
HPGD P15428 3/20 0.50
HSD17B10 Q99714 3/20 0.50
LMNA P02545 2/20 0.50
TOP2A P11388 2/20 0.50
TOP2B Q02880 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
MAPT P10636 1/20 0.48
POLB P06746 3/20 0.46
CACNA1F O60840 1/20 0.46
MAPK1 P28482 1/20 0.46
CACNA1D Q01668 1/20 0.46
CACNA1S Q13698 1/20 0.46
CACNA1C Q13936 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10685966 0.91 KCNH2 (0.58) KCNH2HRH3ALDH1A1KDM4EHPGD
SCHEMBL10683412 0.85 KCNH2 (0.47) KCNH2HRH3ALDH1A1KDM4EHPGD
SCHEMBL9501145 0.85 KCNH2 (0.87) KCNH2HRH3ALDH1A1KDM4EHPGD
SCHEMBL8111734 0.84 KCNH2 (0.71) KCNH2HRH3ALDH1A1KDM4EHPGD
SCHEMBL9501344 0.84 KCNH2 (0.62) KCNH2HRH3ALDH1A1KDM4EHPGD
SCHEMBL9501123 0.84 KDM4E (0.70) KCNH2HRH3ALDH1A1KDM4EHPGD
SCHEMBL9502534 0.83 KCNH2 (0.69) KCNH2HRH3ALDH1A1KDM4EHPGD
SCHEMBL9735289 0.83 KDM4E (0.72) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL9502038 0.83 KCNH2 (0.69) KCNH2HRH3ALDH1A1KDM4EHPGD
SCHEMBL9734255 0.83 KDM4E (0.72) ALDH1A1KDM4EHPGDHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0284935-A1 5-Substituted quinolone- and naphthyridone carboxylic acid derivatives BAYER AG (DE) 1988-10-05 EP claimed
EP-0284935-A1 5-Substituted quinolone- and naphthyridone carboxylic acid derivatives BAYER AG (DE) 1988-10-05 EP disclosed