SCHEMBL9501344

SCHEMBL9501344

CN1CCN(c2cc3c(c(F)c2F)c(=O)c(C(=O)O)cn3C2CC2)CC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.62
HRH3 Q9Y5N1 1/20 0.62
ALDH1A1 P00352 5/20 0.57
KDM4E B2RXH2 4/20 0.57
LMNA P02545 3/20 0.56
HPGD P15428 3/20 0.56
HSD17B10 Q99714 2/20 0.56
MAPT P10636 1/20 0.56
TOP2A P11388 2/20 0.53
TOP2B Q02880 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C9 P11712 1/20 0.53
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
DRD3 P35462 1/20 0.49
PIK3CG P48736 5/20 0.49
PIK3CD O00329 3/20 0.49
PIK3R1 P27986 3/20 0.49
PIK3CA P42336 3/20 0.49
CACNA1F O60840 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556904 0.92 KCNH2 (0.71) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL9501155 0.91 KCNH2 (0.57) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL9504102 0.87 KCNH2 (0.58) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL9501123 0.87 KDM4E (0.70) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL9502038 0.84 KCNH2 (0.69) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL10683407 0.84 KCNH2 (0.64) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL9502534 0.84 KCNH2 (0.69) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL9501145 0.83 KCNH2 (0.87) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL9504545 0.83 KCNH2 (0.63) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL2780752 0.83 ALDH1A1 (0.81) ALDH1A1KDM4ELMNAHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0312085-B1 NOVEL QUINOLINE DERIVATIVES, PROCESSES FOR PREPARATION THEREOF AND ANTIBACTERIAL AGENT CONTAINING THEM Dainippon Pharmaceutical Co., Ltd. (JP) 1993-05-12 EP disclosed
US-5164392-A Active against streptococci and staphylococci DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1992-11-17 US disclosed
US-5013841-A Oxo quinoline derivatives DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1991-05-07 US disclosed
EP-0312085-A2 Novel quinoline derivatives, processes for preparation thereof and antibacterial agent containing them Dainippon Pharmaceutical Co., Ltd. (JP) 1989-04-19 EP disclosed