SCHEMBL10685404

SCHEMBL10685404

O=C(O)CCCSc1ccc(C(=O)O)cn1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 5/20 0.64
CXCR1 P25024 3/20 0.64
ALDH1A1 P00352 3/20 0.57
CYP1A2 P05177 1/20 0.57
CYP2C9 P11712 1/20 0.57
HPGD P15428 1/20 0.57
CYP2C19 P33261 1/20 0.57
HSD17B10 Q99714 1/20 0.57
TP53 P04637 1/20 0.45
P4HA1 P13674 2/20 0.44
P4HTM Q9NXG6 2/20 0.44
KDM4E B2RXH2 2/20 0.44
MIF P14174 1/20 0.43
GABRP O00591 1/20 0.42
GABRD O14764 1/20 0.42
GABRA1 P14867 1/20 0.42
GABRB1 P18505 1/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA5 P31644 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12863439 0.85 ALDH1A1 (0.63) CXCR2CXCR1ALDH1A1CYP1A2CYP2C9
SCHEMBL839476 0.84 ALDH1A1 (0.57) CXCR2CXCR1ALDH1A1CYP1A2CYP2C9
SCHEMBL5445067 0.80 ALDH1A1 (0.65) CXCR2CXCR1ALDH1A1CYP1A2CYP2C9
SCHEMBL5846781 0.79 CXCR2 (1.00) CXCR2CXCR1KDM4E
SCHEMBL796738 0.78 ALDH1A1 (0.57) CXCR2CXCR1ALDH1A1CYP1A2CYP2C9
SCHEMBL417669 0.78 ALDH1A1 (0.57) CXCR2CXCR1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL16456689 0.78 CXCR1 (0.51) CXCR2CXCR1ALDH1A1CYP1A2CYP2C9
SCHEMBL4432631 0.77 ALDH1A1 (0.65) ALDH1A1CYP1A2CYP2C9HPGDCYP2C19
SCHEMBL796408 0.74 ALDH1A1 (0.61) CXCR2CXCR1ALDH1A1CYP1A2CYP2C9
SCHEMBL13787819 0.74 ALDH1A1 (0.61) CXCR2ALDH1A1CYP1A2CYP2C9HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4762848-A IMMUNE SYSTEM STIMULANTS, CYTOSTATIC AGENTS HOECHST AKTIENGESELLSCHAFT (DE) 1988-08-09 US disclosed
EP-0194572-A1 Heterocyclic sulfides, process for their preparation and Medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1986-09-17 EP disclosed