SCHEMBL10685652

SCHEMBL10685652

CC(CO)(CO)NCc1cccc2c(Cl)c3ccccc3cc12

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.42
CD274 Q9NZQ7 6/20 0.36
PDCD1 Q15116 4/20 0.35
PDCD1LG2 Q9BQ51 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
MAPT P10636 1/20 0.34
PKM P14618 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
MAPK1 P28482 1/20 0.33
MC5R P33032 1/20 0.33
NPBWR1 P48145 1/20 0.33
MCHR1 Q99705 1/20 0.33
HPGD P15428 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10488341 0.94 SLC2A1 (0.50) SLC2A1CD274PDCD1CYP1A2CYP3A4
SCHEMBL10488864 0.85 SLC2A1 (0.46) SLC2A1CD274PDCD1MAPTKMT2A
SCHEMBL10488906 0.84 SLC2A1 (0.42) SLC2A1CD274PDCD1MAPTKMT2A
Hydrochloric Acid SCHEMBL10488204 0.83 SLC2A1 (0.45) SLC2A1CD274PDCD1MAPTKMT2A
Hydrochloric Acid SCHEMBL10488254 0.83 SLC2A1 (0.41) SLC2A1CD274PDCD1MAPTKMT2A
SCHEMBL10803667 0.80 NPBWR1 (0.35) SLC2A1CD274KMT2ANPBWR1MCHR1
SCHEMBL10349041 0.80 NPBWR1 (0.38) SLC2A1CD274CYP1A2KMT2ANPBWR1
SCHEMBL11091727 0.80 KMT2A (0.34) CD274PDCD1LG2CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL10349542 0.79 NPBWR1 (0.40) SLC2A1CD274CYP1A2KMT2ANPBWR1
SCHEMBL9466408 0.78 SLC2A1 (0.38) SLC2A1CD274PDCD1CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0125702-B1 POLYCYCLIC AROMATIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1987-08-12 EP claimed
EP-0125702-A2 Polycyclic aromatic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-21 EP claimed
US-4719049-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1988-01-12 US disclosed
EP-0125702-A2 Polycyclic aromatic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1984-11-21 EP disclosed