SCHEMBL10690001

SCHEMBL10690001

COC(=O)CNC(=O)C(Cc1ccccc1)C(=O)NOCc1ccccc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MME P08473 1/20 0.53
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
ABCC3 O15438 1/20 0.48
NR1I2 O75469 1/20 0.48
ABCB11 O95342 1/20 0.48
NR3C1 P04150 1/20 0.48
RARG P13631 1/20 0.48
CNR1 P21554 1/20 0.48
OPRK1 P41145 1/20 0.48
NR1H2 P55055 1/20 0.48
PPARA Q07869 1/20 0.48
NR1H3 Q13133 1/20 0.48
NR1I3 Q14994 1/20 0.48
MMP8 P22894 3/20 0.48
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10691292 0.90 CYP1A2 (0.57) MMECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL10692309 0.88 MME (0.69) MMEMMP8NPC1RAB9A
SCHEMBL10687449 0.85 MME (0.74) MMEMMP8
SCHEMBL1258101 0.81 NPC1 (0.57) MMECYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL10686998 0.81 LAP3 (0.51) MMEMMP8
SCHEMBL6162382 0.79 SLC7A5 (0.53) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7635307 0.79 SLC7A5 (0.53) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL11202440 0.78 SLC7A5 (0.51) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL11202436 0.78 SLC7A5 (0.51) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL11940451 0.77 CYP3A4 (0.63) MMECYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4738803-A ENZYME INHIBITORS ROQUES BERNARD (FR) 1988-04-19 US disclosed
US-4618708-A ENKEPHALINASE INHIBITOR, ANALGESICS, ANTIDEPRESSANT, ANTIDIARRHEA, OR HYPOTENSIVE AGENT ROQUES BERNARD (FR) 1986-10-21 US disclosed