SCHEMBL10690417

SCHEMBL10690417

COc1cc(N2C3CCC2CC(c2c(N)nc(N)nc2Cl)C3)cc(OC)c1OC

nearest known ligand 0.47

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10689261 0.86 FGFR1 (0.33)
SCHEMBL10687474 0.82 NEK2 (0.40) HSP90AA1HSP90AB1
SCHEMBL10689477 0.82 DHFR (0.39)
SCHEMBL10691189 0.81 DHFR (0.40) HSP90AA1HSP90AB1
SCHEMBL10687469 0.80 HSP90AA1 (0.39) HSP90AA1HSP90AB1
SCHEMBL10687297 0.79 DHFR (0.47)
SCHEMBL10803047 0.76 GAA (0.42)
SCHEMBL8207060 0.68 DHFR (0.36)
SCHEMBL10687594 0.68 SMN1; SMN2 (0.41)
SCHEMBL10687580 0.67 MEN1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4774249-A Pyrimidine derivatives for treating malaria HOFFMANN-LA ROCHE INC. (US) 1988-09-27 US disclosed
EP-0122580-B1 PYRIMIDINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1987-10-28 EP disclosed
US-4590270-A 2,4-diamino-[4-piperidinyl]pyrimidines useful as antibacterial agents, antimalarial agents, antitumors agents HOFFMANN-LA ROCHE INC. (US) 1986-05-20 US disclosed
EP-0122580-A1 Pyrimidine derivatives, their preparation and pharmaceutical compositions F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1984-10-24 EP disclosed