SCHEMBL10690764

SCHEMBL10690764

Nc1ncc(C2CCN(c3ccc(Cl)cc3)CC2)c(N)n1

nearest known ligand 0.71

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DHFR P00374 14/20 0.63
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10686944 0.83 DHFR (0.45) DHFR
SCHEMBL10691450 0.83 DHFR (0.65) DHFR
SCHEMBL10690355 0.81 MEN1 (0.54) DHFR
SCHEMBL20734745 0.79 DHFR (0.67) DHFR
SCHEMBL10689416 0.78 DHFR (0.52) DHFR
SCHEMBL20804285 0.77 DHFR (1.00) DHFR
SCHEMBL20734741 0.76 DHFR (0.50) DHFR
SCHEMBL10807304 0.76 DHFR (0.56) DHFR
SCHEMBL2444528 0.75 DHFR (0.41) DHFR
SCHEMBL30714999 0.75 DHFR (0.41) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0122580-B1 PYRIMIDINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1987-10-28 EP claimed
US-4590270-A 2,4-diamino-[4-piperidinyl]pyrimidines useful as antibacterial agents, antimalarial agents, antitumors agents HOFFMANN-LA ROCHE INC. (US) 1986-05-20 US claimed
EP-0122580-A1 Pyrimidine derivatives, their preparation and pharmaceutical compositions F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1984-10-24 EP claimed
US-4774249-A Pyrimidine derivatives for treating malaria HOFFMANN-LA ROCHE INC. (US) 1988-09-27 US disclosed
EP-0122580-B1 PYRIMIDINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1987-10-28 EP disclosed
US-4590270-A 2,4-diamino-[4-piperidinyl]pyrimidines useful as antibacterial agents, antimalarial agents, antitumors agents HOFFMANN-LA ROCHE INC. (US) 1986-05-20 US disclosed