SCHEMBL10690794

SCHEMBL10690794

C=CCCN1C(C)=C(C(=O)OCC)C(c2ccc(C(F)(F)F)cc2)C(C(=O)OCC)=C1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.49
HPGD P15428 3/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
KDM4E B2RXH2 4/20 0.48
GAA P10253 2/20 0.48
HTT P42858 1/20 0.47
CYP3A4 P08684 3/20 0.43
ELANE P08246 2/20 0.43
CYP2C9 P11712 2/20 0.43
ATM Q13315 1/20 0.43
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
PTPN1 P18031 1/20 0.41
TSHR P16473 3/20 0.41
ALDH1A1 P00352 3/20 0.40
GPBAR1 Q8TDU6 1/20 0.40
ABCC1 P33527 1/20 0.39
HSD17B10 Q99714 2/20 0.39
TP53 P04637 1/20 0.39
ACHE P22303 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836701 0.87 KMT2A (0.49) NPSR1KDM4EGAACYP3A4ELANE
SCHEMBL9120147 0.83 NPSR1 (0.69) NPSR1HPGDSMN1; SMN2KDM4EGAA
SCHEMBL11818486 0.80 SMN1; SMN2 (0.53) NPSR1HPGDSMN1; SMN2KDM4EGAA
SCHEMBL21116053 0.79 HTT (0.71) NPSR1HPGDSMN1; SMN2KDM4EGAA
SCHEMBL7492934 0.78 HSP90AA1 (0.56) NPSR1HPGDSMN1; SMN2KDM4EGAA
SCHEMBL9120841 0.77 KDM4E (0.51) NPSR1HPGDSMN1; SMN2KDM4EGAA
SCHEMBL9118463 0.75 HSP90AA1 (0.55) NPSR1HPGDKDM4EGAAHTT
SCHEMBL11820276 0.74 KDM4E (0.70) HPGDSMN1; SMN2KDM4EGAACYP3A4
SCHEMBL9836195 0.74 LMNA (0.53) NPSR1HPGDKDM4EGAATSHR
SCHEMBL7431402 0.73 HSP90AA1 (0.42) NPSR1HPGDSMN1; SMN2KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4721708-A CYCLICATION WITH LEWIS ACIDS MERCK & CO., INC. (US) 1988-01-26 US disclosed