SCHEMBL10691398

SCHEMBL10691398

C=CNC=CCCCCC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.46
FAAH O00519 2/20 0.41
TRPV1 Q8NER1 2/20 0.41
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.37
CYP3A4 P08684 1/20 0.37
KMT2A Q03164 1/20 0.37
GMNN O75496 1/20 0.36
USP2 O75604 1/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36
APEX1 P27695 1/20 0.36
CYP2C19 P33261 1/20 0.36
RECQL P46063 1/20 0.36
BLM P54132 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9630645 0.98 TSHR (0.50) TSHRFAAHTRPV1MEN1CYP3A4
SCHEMBL9630640 0.98 TSHR (0.50) TSHRFAAHTRPV1MEN1CYP3A4
SCHEMBL1485910 0.93
SCHEMBL1485908 0.93
SCHEMBL284503 0.85 FAAH (0.48) TSHRFAAHTRPV1ALDH1A1MEN1
SCHEMBL284502 0.85 FAAH (0.48) TSHRFAAHTRPV1ALDH1A1MEN1
SCHEMBL7103122 0.83 FAAH (0.52) TSHRFAAHTRPV1MEN1CYP3A4
SCHEMBL1485591 0.83
SCHEMBL22015838 0.83 FAAH (0.52) TSHRFAAHTRPV1MEN1CYP3A4
SCHEMBL8699327 0.83 FAAH (0.52) TSHRFAAHTRPV1MEN1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4760089-A Benzonitrile derivative; enzyme inhibitor SMITHKLINE BECKMAN CORPORATION (US) 1988-07-26 US disclosed
EP-0219961-A1 Irreversible dopamine-B-hydroxylase inhibitors SMITHKLINE BECKMAN CORPORATION (US) 1987-04-29 EP disclosed