SCHEMBL10691807

SCHEMBL10691807

CCOc1cc2cc(C(=O)N(CC)CC)sc2cc1OCC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
KMT2A Q03164 1/20 0.53
STING1 Q86WV6 14/20 0.47
TRPM8 Q7Z2W7 1/20 0.44
ALDH1A1 P00352 2/20 0.43
GLA P06280 2/20 0.43
NPC1 O15118 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
ALOX12 P18054 1/20 0.43
RAB9A P51151 1/20 0.43
CLK1 P49759 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tibenelast SCHEMBL449748 0.82 STING1 (0.54) HPGDSTING1ALDH1A1TSHR
SCHEMBL10688443 0.81 STING1 (0.53) STING1TSHRCLK1HDAC3HDAC4
Tibenelast SCHEMBL635433 0.81 STING1 (0.53) HPGDSTING1ALDH1A1TSHR
SCHEMBL10692662 0.81 STING1 (0.50) STING1TSHRCLK1HDAC3HDAC4
Tibenelast SCHEMBL10688452 0.81 STING1 (0.53) HPGDSTING1ALDH1A1TSHR
Tibenelast SCHEMBL635432 0.79 STING1 (0.49) STING1CLK1HDAC3HDAC4HDAC1
SCHEMBL10642176 0.77 STING1 (0.60) STING1
SCHEMBL10641965 0.77 STING1 (0.60) STING1
SCHEMBL10537567 0.76 STING1 (0.49) HPGDSTING1ALDH1A1TSHRCLK1
SCHEMBL10534791 0.76 STING1 (0.49) HPGDSTING1ALDH1A1TSHRCLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0253650-A2 Improvements relating to benzothiophene derivatives ELI LILLY AND COMPANY (US) 1988-01-20 EP disclosed