SCHEMBL10692858

SCHEMBL10692858

O=C(O)c1cn(C2CC2)c2c(Cl)c(N3CCC(CNCCF)C3)c(F)cc2c1=O

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.69
POLB P06746 3/20 0.69
OPRM1 P35372 2/20 0.69
CHRM2 P08172 1/20 0.69
CHRM1 P11229 1/20 0.69
OPRD1 P41143 1/20 0.69
KCNH2 Q12809 7/20 0.61
KDM4E B2RXH2 5/20 0.49
HPGD P15428 3/20 0.49
TDP1 Q9NUW8 2/20 0.49
PRKD3 O94806 1/20 0.49
ALOX15 P16050 1/20 0.49
CLK2 P49760 1/20 0.49
HSD17B10 Q99714 1/20 0.49
CLK4 Q9HAZ1 1/20 0.49
LMNA P02545 2/20 0.47
NPSR1 Q6W5P4 1/20 0.46
TOP1 P11387 2/20 0.45
TOP2A P11388 2/20 0.44
TOP2B Q02880 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10762411 0.93 ALDH1A1 (0.69) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10692692 0.91 KCNH2 (0.65) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10530714 0.91 ALDH1A1 (0.70) ALDH1A1POLBOPRM1CHRM2CHRM1
Hydrochloric Acid SCHEMBL10529374 0.89 ALDH1A1 (0.70) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL5571239 0.89 ALDH1A1 (0.78) ALDH1A1POLBOPRM1CHRM2CHRM1
Hydrochloric Acid SCHEMBL10530738 0.88 ALDH1A1 (0.77) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9733802 0.88 ALDH1A1 (0.76) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL6489034 0.88 ALDH1A1 (0.76) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9734892 0.88 ALDH1A1 (0.76) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10764195 0.84 KCNH2 (0.63) ALDH1A1POLBOPRM1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4791118-A BACTERICIDES; GRAMNEGATIVE AND -POSITIVE BACTERIA; ANIMAL INFECTIONS; PLANT DISEASES KYORIN PHARMACEUTICAL CO., LTD. (JP) 1988-12-13 US claimed
US-4791118-A BACTERICIDES; GRAMNEGATIVE AND -POSITIVE BACTERIA; ANIMAL INFECTIONS; PLANT DISEASES KYORIN PHARMACEUTICAL CO., LTD. (JP) 1988-12-13 US disclosed
EP-0216323-A2 Quinolonecarboxylic acid derivatives and their preparation KYORIN PHARMACEUTICAL CO., LTD. (JP) 1987-04-01 EP disclosed