SCHEMBL10692951

SCHEMBL10692951

COC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1cc([N+](=O)[O-])ccc1OCCBr

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.53
MAPT P10636 5/20 0.53
HIF1A Q16665 4/20 0.53
KMT2A Q03164 4/20 0.53
CYP1A2 P05177 3/20 0.53
CYP3A4 P08684 3/20 0.53
CYP2C9 P11712 3/20 0.53
CYP2C19 P33261 3/20 0.53
MEN1 O00255 3/20 0.53
LMNA P02545 2/20 0.53
MAPK1 P28482 2/20 0.53
CYP2D6 P10635 2/20 0.53
TSHR P16473 2/20 0.53
NFKB1 P19838 2/20 0.53
THPO P40225 2/20 0.53
CACNA1C Q13936 2/20 0.53
POLB P06746 1/20 0.53
GPR55 Q9Y2T6 1/20 0.53
TDP1 Q9NUW8 3/20 0.52
KDM4E B2RXH2 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9789920 0.94 ADORA3 (0.52) ADORA3MAPTHIF1AKMT2ACYP1A2
SCHEMBL9825000 0.91 ADORA3 (0.54) ADORA3MAPTHIF1AKMT2ACYP1A2
SCHEMBL10488517 0.90 ADORA3 (0.53) ADORA3MAPTHIF1AKMT2ACYP1A2
SCHEMBL7406051 0.89 ADORA3 (0.53) ADORA3MAPTHIF1AKMT2ACYP1A2
SCHEMBL10488355 0.89 ADORA3 (0.53) ADORA3MAPTHIF1AKMT2ACYP1A2
SCHEMBL7287257 0.89 ADORA3 (0.53) ADORA3MAPTHIF1AKMT2ACYP1A2
SCHEMBL9485672 0.88 ADORA3 (0.53) ADORA3MAPTHIF1AKMT2ACYP1A2
SCHEMBL7400745 0.86 ADORA3 (0.55) ADORA3MAPTHIF1AKMT2ACYP1A2
Hydrochloric Acid SCHEMBL7276770 0.86 ADORA3 (0.50) ADORA3MAPTHIF1AKMT2ACYP1A2
SCHEMBL7396515 0.85 ADORA3 (0.43) ADORA3MAPTHIF1AKMT2ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4727082-A CARDIOVASCULAR DISORDERS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1988-02-23 US disclosed
EP-0167371-A2 Dihydropyridine compounds, their production, and pharmaceutical compositions containing them YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1986-01-08 EP disclosed