SCHEMBL10693042

SCHEMBL10693042

CC1(N)Cc2ccccc2NC1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 2/20 0.46
AHR P35869 1/20 0.46
BRD4 O60885 3/20 0.44
CREBBP Q92793 2/20 0.44
NPC1 O15118 2/20 0.44
MAPK13 O15264 1/20 0.44
MAPK12 P53778 1/20 0.44
MAPK11 Q15759 1/20 0.44
MAPK14 Q16539 1/20 0.44
PDK4 Q16654 1/20 0.44
OTUD7B Q6GQQ9 1/20 0.42
MAPT P10636 3/20 0.42
HTR5A P47898 4/20 0.38
SRC P12931 1/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
HSP90AA1 P07900 1/20 0.37
THRB P10828 1/20 0.37
HK1 P19367 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30100699 0.81 PDK2 (0.48) PDK2AHRBRD4CREBBPNPC1
SCHEMBL6220027 0.81 PDK2 (0.48) PDK2AHRBRD4CREBBPNPC1
SCHEMBL23674847 0.75 NPSR1 (0.52) PDK2AHRBRD4CREBBPNPC1
SCHEMBL30100714 0.75 NPSR1 (0.52) PDK2AHRBRD4CREBBPNPC1
SCHEMBL13090519 0.74 MAPT (0.42) PDK2AHRBRD4CREBBPNPC1
SCHEMBL9194873 0.74 PDK2 (0.42) PDK2AHRBRD4CREBBPNPC1
SCHEMBL14941425 0.73 OTUD7B (0.59) PDK2AHRBRD4CREBBPNPC1
SCHEMBL30293249 0.73 OTUD7B (0.59) PDK2AHRBRD4CREBBPNPC1
SCHEMBL28394080 0.73 PDK2 (0.48) PDK2AHRBRD4CREBBPNPC1
SCHEMBL8524680 0.72 AHR (0.57) PDK2AHRBRD4CREBBPNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4757068-A Lactams and bicyclic lactams useful as cholecystokinin antagonists MERCK & CO., INC. (US) 1988-07-12 US disclosed