SCHEMBL10693832

SCHEMBL10693832

COC(=O)c1ccc2c(c1)C(c1ccccc1)=NCC(=O)N2

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 2/20 0.61
CNR1 P21554 1/20 0.61
NTSR1 P30989 1/20 0.61
OPRK1 P41145 1/20 0.61
GABRA1 P14867 4/20 0.59
GABRA5 P31644 4/20 0.59
GABRA3 P34903 4/20 0.59
GABRA2 P47869 4/20 0.59
GABRB2 P47870 4/20 0.59
GABRG2 P18507 2/20 0.59
GABRB3 P28472 2/20 0.59
LMNA P02545 3/20 0.57
HPGD P15428 1/20 0.57
KMT2A Q03164 1/20 0.51
CCNB2 O95067 1/20 0.47
CDK1 P06493 1/20 0.47
CCNB1 P14635 1/20 0.47
MDH2 P40926 1/20 0.47
GSK3B P49841 1/20 0.47
CCNB3 Q8WWL7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9654320 0.85 GABRA1 (0.66) PDE4DCNR1NTSR1OPRK1GABRA1
SCHEMBL4709615 0.81 PDE4D (0.67) PDE4DCNR1NTSR1OPRK1GABRA1
SCHEMBL11821347 0.79 CHRM1 (0.71) PDE4DCNR1NTSR1OPRK1GABRA1
SCHEMBL11776007 0.78 PDE4D (0.70) PDE4DCNR1NTSR1OPRK1GABRA1
SCHEMBL15198055 0.78 EGFR (0.50) GABRA5GABRA3GABRG2GABRB3HPGD
SCHEMBL9654207 0.77 PDE4D (0.61) PDE4DCNR1NTSR1OPRK1GABRA1
SCHEMBL5349947 0.77 GABRA1 (0.62) PDE4DCNR1NTSR1OPRK1GABRA1
SCHEMBL1421181 0.76 KMT2A (0.82) PDE4DCNR1NTSR1OPRK1GABRA1
SCHEMBL13538415 0.76 PDE4D (0.71) PDE4DCNR1NTSR1OPRK1GABRA1
Ro-053061 SCHEMBL2615407 0.76 PDE4D (0.71) PDE4DCNR1NTSR1OPRK1GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0255028-A2 1,4-Benzodiazepines, their preparation and use as PAF antagonists BOEHRINGER INGELHEIM KG (DE) 1988-02-03 EP disclosed