SCHEMBL10695935

SCHEMBL10695935

CCCCCN1C(=O)C(C)(C)c2cc3nc(-c4coc(C)c4)[nH]c3cc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 3/20 0.48
AURKB Q96GD4 3/20 0.48
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
TSSK1B Q9BXA7 1/20 0.33
MEN1 O00255 5/20 0.33
KMT2A Q03164 5/20 0.33
SCN9A Q15858 4/20 0.32
BRD4 O60885 1/20 0.32
CHEK1 O14757 1/20 0.32
SRC P12931 1/20 0.32
CDK2 P24941 1/20 0.32
KDR P35968 1/20 0.32
FLT3 P36888 1/20 0.32
GSK3B P49841 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10701072 0.90 AURKA (0.59) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10698460 0.86 AURKA (0.48) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10695107 0.86 AURKA (0.46) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10693690 0.84 PDE4A (0.51) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10695197 0.82 AURKA (0.46) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10695207 0.82 AURKB (0.46) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10696394 0.81 PDE4A (0.52) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL13368132 0.81 AURKA (0.53) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10695285 0.81 AURKA (0.47) AURKAAURKB
SCHEMBL13341481 0.81 AURKA (0.45) AURKAAURKBPDE3BPDE3AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed