SCHEMBL10698460

SCHEMBL10698460

COCCN1C(=O)C(C)(C)c2cc3nc(-c4coc(C)c4)[nH]c3cc21

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AURKA O14965 3/20 0.48
AURKB Q96GD4 3/20 0.48
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
BRD4 O60885 1/20 0.31
RHEB Q15382 1/20 0.30
AMY1A P0DUB6 1/20 0.30
CHEK1 O14757 1/20 0.30
SRC P12931 1/20 0.30
CDK2 P24941 1/20 0.30
KDR P35968 1/20 0.30
FLT3 P36888 1/20 0.30
GSK3B P49841 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10701072 0.88 AURKA (0.59) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10695935 0.86 AURKA (0.48) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10699944 0.86 AURKA (0.46) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10698025 0.84 PDE4A (0.51) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10700270 0.83 AURKA (0.47) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10698967 0.83 AURKB (0.47) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10698233 0.82 AURKA (0.46) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL4143677 0.82 AURKA (0.73) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10698273 0.81 MAPT (0.47) AURKAAURKBPDE4APDE4BPDE4C
SCHEMBL10696985 0.80 AURKA (0.40) AURKAAURKBPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed