SCHEMBL10696958

SCHEMBL10696958

CN1CCN(c2c(F)cc3c(=O)c(C(=O)O)cn(C4CC4)c3c2Cl)CC1c1cccs1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.62
POLB P06746 3/20 0.62
OPRM1 P35372 2/20 0.62
CHRM2 P08172 1/20 0.62
CHRM1 P11229 1/20 0.62
OPRD1 P41143 1/20 0.62
KCNH2 Q12809 5/20 0.49
KDM4E B2RXH2 10/20 0.48
HPGD P15428 5/20 0.48
HSD17B10 Q99714 3/20 0.48
TDP1 Q9NUW8 2/20 0.48
PRKD3 O94806 1/20 0.48
ALOX15 P16050 1/20 0.48
CLK2 P49760 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48
LMNA P02545 2/20 0.46
NPSR1 Q6W5P4 1/20 0.45
TOP2A P11388 1/20 0.45
TOP2B Q02880 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8434019 0.84 ALDH1A1 (0.62) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10695310 0.83 ALDH1A1 (0.70) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10640499 0.83 ALDH1A1 (0.49) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL312998 0.82 ALDH1A1 (0.72) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10510158 0.79 KCNH2 (0.46) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL26194819 0.79 ALDH1A1 (0.79) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9671640 0.79 ALDH1A1 (0.72) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL29055626 0.79 ALDH1A1 (0.73) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL10636991 0.78 ALDH1A1 (0.59) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9734537 0.78 ALDH1A1 (0.80) ALDH1A1POLBOPRM1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0264050-A2 7-Amino-1-cyclopropyl-8-chloro-6-fluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids, process for their preparation and antibacterial agents containing them BAYER AG (DE) 1988-04-20 EP disclosed