SCHEMBL10697156

SCHEMBL10697156

Nc1ccc(Cc2ncc[nH]2)cc1N

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 8/20 0.56
HTR1A P08908 1/20 0.41
CYP17A1 P05093 1/20 0.40
CYP19A1 P11511 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
ALOX15 P16050 1/20 0.37
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
CYP3A4 P08684 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7726175 0.82 TAAR1 (0.47) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL13372830 0.81 TAAR1 (0.80) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL177767 0.80 TAAR1 (0.67) TAAR1HTR1ACYP17A1CYP19A1CYP11B1
SCHEMBL31414967 0.78 TAAR1 (0.75) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL10463711 0.78 TAAR1 (0.64) TAAR1HTR1ACYP19A1CYP11B1CYP11B2
SCHEMBL11295655 0.77 TAAR1 (0.58) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL27582729 0.75 TAAR1 (0.64) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL11295562 0.74 TAAR1 (0.69) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL508430 0.73 TAAR1 (0.53) TAAR1HTR1ACYP17A1CYP11B1CYP11B2
SCHEMBL10679401 0.73 TAAR1 (0.53) TAAR1HTR1AADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0260744-A2 (1H-imidazol-1-ylmethyl) substituted benzimidazole derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1988-03-23 EP disclosed