SCHEMBL11295655

SCHEMBL11295655

Cc1ccc(Cc2ncc[nH]2)cc1C

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 11/20 0.58
HTR1A P08908 1/20 0.46
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
ALOX15 P16050 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
BRD4 O60885 1/20 0.36
LMNA P02545 1/20 0.36
GLA P06280 1/20 0.36
BLM P54132 1/20 0.36
PMP22 Q01453 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11288699 0.86 TAAR1 (0.46) TAAR1HTR1AALOX15SMN1; SMN2ALDH1A1
SCHEMBL13372830 0.82 TAAR1 (0.80) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL11290757 0.82 TBXAS1 (0.48) TAAR1HTR1AALOX15
SCHEMBL11295562 0.79 TAAR1 (0.69) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL31414967 0.79 TAAR1 (0.75) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL11290384 0.78 TAAR1 (0.67) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL10719843 0.77 TAAR1 (0.66) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL10697156 0.77 TAAR1 (0.56) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL954941 0.76 TAAR1 (0.54) TAAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL27582729 0.76 TAAR1 (0.64) TAAR1HTR1AADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0003732-A2 Imidazole derivatives and salts thereof, their synthesis, and pharmaceutical formulations thereof THE WELLCOME FOUNDATION LIMITED (GB) 1979-09-05 EP claimed
EP-0064820-A1 Substituted imidazole and imidazoline derivatives and their preparation and use Farmos-Yhtyma Oy (FI) 1982-11-17 EP disclosed