SCHEMBL10708448

SCHEMBL10708448

CCN1C(=O)C(C)(C)c2cc(NC(=O)c3ccc(Cl)cc3)c([N+](=O)[O-])cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 1/20 0.47
MAPT P10636 6/20 0.45
GAA P10253 2/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TP53 P04637 2/20 0.41
POLB P06746 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
CPT2 P23786 1/20 0.40
CPT1A P50416 1/20 0.40
CPT1B Q92523 1/20 0.40
LMNA P02545 2/20 0.40
MAPK1 P28482 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
HCAR3 P49019 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2485998 0.92 MAPT (0.46) PHGDHMAPTGAAHTTNPSR1
SCHEMBL10714574 0.90 MAPT (0.40) MAPTGAAHTTTP53NPC1
SCHEMBL10711637 0.90 NPC1 (0.48) MAPTGAAHTTNPSR1POLB
SCHEMBL10700306 0.89 MAPT (0.51) MAPTGAAPOLBNPC1RAB9A
SCHEMBL10711757 0.89 MAPT (0.40) MAPTGAAHTTNPC1RAB9A
SCHEMBL10709119 0.89 MAPT (0.41) MAPTGAAHTTPOLBNPC1
SCHEMBL10704419 0.89 MAPT (0.41) MAPTGAAHTTNPSR1NPC1
SCHEMBL10711705 0.87 AURKA (0.36) MAPTGAAHTTNPSR1TP53
SCHEMBL10710846 0.87 TP53 (0.35) MAPTGAAHTTNPSR1TP53
SCHEMBL2516093 0.86 HTT (0.39) MAPTGAAHTTNPSR1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268178-A1 Pyrrolo-benzimidazoles, medicaments containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1988-05-25 EP disclosed