SCHEMBL10714404

SCHEMBL10714404

Nc1cccc(C(F)(F)C(F)(F)c2cccc(N)c2)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.74
MAPK1 P28482 1/20 0.74
CYP3A4 P08684 2/20 0.52
CASP1 P29466 1/20 0.52
RECQL P46063 1/20 0.52
ALDH1A1 P00352 4/20 0.42
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
CA14 Q9ULX7 2/20 0.42
CA7 P43166 1/20 0.42
PTGS1 P23219 3/20 0.41
MAOA P21397 3/20 0.41
LMNA P02545 2/20 0.38
GAA P10253 2/20 0.38
KDM4E B2RXH2 2/20 0.38
GLA P06280 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3843446 0.91 TSHR (0.68) TSHRMAPK1CYP3A4CASP1RECQL
SCHEMBL29402206 0.91 TSHR (0.68) TSHRMAPK1CYP3A4CASP1RECQL
SCHEMBL3867382 0.91 TSHR (0.68) TSHRMAPK1CYP3A4CASP1RECQL
SCHEMBL29405287 0.89 TSHR (0.65) TSHRMAPK1CYP3A4CASP1RECQL
SCHEMBL8974219 0.89 TSHR (0.65) TSHRMAPK1CYP3A4CASP1RECQL
SCHEMBL8167656 0.87 TSHR (0.63) TSHRMAPK1CYP3A4CASP1RECQL
SCHEMBL7586287 0.87 TSHR (0.63) TSHRMAPK1CYP3A4CASP1RECQL
SCHEMBL125470 0.85 TSHR (0.74) TSHRMAPK1CYP3A4CASP1RECQL
SCHEMBL29410732 0.85 TSHR (1.00) TSHRMAPK1CYP3A4CASP1RECQL
SCHEMBL39591 0.85 TSHR (1.00) TSHRMAPK1CYP3A4CASP1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0201778-B1 (METH)-ACRYLIC-ACID ESTERS AND THEIR USE BAYER AG (DE) 1988-12-28 EP disclosed
EP-0201778-A1 (Meth)-acrylic-acid esters and their use BAYER AG (DE) 1986-11-20 EP disclosed