SCHEMBL10715411

SCHEMBL10715411

COc1c(C)cnc(CSc2nc3cscc3[nH]2)c1C

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRS3 P32247 3/20 0.68
SHMT2 P34897 1/20 0.44
AGXT P21549 1/20 0.42
KMT2A Q03164 4/20 0.42
WDR5 P61964 3/20 0.42
CYP2C9 P11712 5/20 0.40
CYP1A2 P05177 4/20 0.40
CYP3A4 P08684 4/20 0.40
CYP2C19 P33261 4/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
ATP4A P20648 3/20 0.40
ATP4B P51164 3/20 0.40
DDAH1 O94760 2/20 0.40
ENGASE Q8NFI3 2/20 0.40
HTT P42858 2/20 0.40
ATP1A1 P05023 2/20 0.40
ATP1B1 P05026 2/20 0.40
ATP1A3 P13637 2/20 0.40
ATP1B2 P14415 2/20 0.40
ATP1A2 P50993 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10578851 0.84 BRS3 (0.74) BRS3SHMT2KMT2AWDR5CYP2C9
Ufiprazole SCHEMBL1816535 0.81 BRS3 (1.00) BRS3KMT2AWDR5CYP2C9CYP1A2
Ufiprazole SCHEMBL29693729 0.81 BRS3 (1.00) BRS3KMT2AWDR5CYP2C9CYP1A2
Ufiprazole SCHEMBL662986 0.81 BRS3 (0.84) BRS3KMT2AWDR5CYP2C9CYP1A2
Ufiprazole SCHEMBL29455226 0.81 BRS3 (0.84) BRS3KMT2AWDR5CYP2C9CYP1A2
Ufiprazole SCHEMBL3180530 0.81 BRS3 (0.76) BRS3SHMT2KMT2AWDR5CYP2C9
SCHEMBL14648553 0.80 BRS3 (0.69) BRS3SHMT2AGXTKMT2AWDR5
Ufiprazole SCHEMBL7929368 0.80 BRS3 (0.82) BRS3KMT2AWDR5CYP2C9CYP1A2
Ufiprazole SCHEMBL31529606 0.80 BRS3 (0.82) BRS3KMT2AWDR5CYP2C9CYP1A2
SCHEMBL19974777 0.80 BRS3 (0.66) BRS3SHMT2AGXTKMT2AWDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1987005296-A1 2-[(2-PYRIDYL)METHYLSULFINYL]THIENOIMIDAZOLES AND RELATED COMPOUNDS AS ANTIULCER AGENTS PFIZER INC. (US) 1987-09-11 WO disclosed